Target Details
UniProt ACQ14289
Gene SymbolPTK2B
Protein NameProtein-tyrosine kinase 2-beta
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF21477 (FERM_C_FAK1) PF00373 (FERM_M) PF18038 (FERM_N_2) PF03623 (Focal_AT) PF07714 (PK_Tyr_Ser-Thr)
Summary
  • Multi-target molecules 210
  • Clinical molecules 15
  • Avg pChEMBL 7.28
Top Co-occurrence Targets
Active Molecules (210)
InChIKey pChEMBL Type Targets Clinical
CEOVOUHGBMXHLJ 9.8 Ki 2
DPRFHIQZBTUOOM 9.7 Ki 2
HPQAVQJTTFEWSN 9.4 Ki 2
FKCIIMYQSRTZNM 9.2 IC50 2
BGNMLKFHDPQLLJ 9.2 IC50 2
VRRYDMZFZWURRY 9.2 Ki 2
NGHZDJWRZKYLSD 9.1 IC50 2
YKEMNGJUZQIQPN 9.0 Ki 2
XZCSQNOUJUIWEB 9.0 Ki 2
QQWUGDVOUVUTOY 9.0 Kd 231 Yes
HMFCBYNYXTWSRZ 8.8 IC50 2
INVLFTRLOIZJTP 8.8 Ki 2
LKQQDFRBWPNRJF 8.8 Ki 2
WFYYQQDXEBYUGQ 8.7 IC50 2
JKXHCHABOHZRIC 8.7 IC50 2
PVJVEBBWSBNEJJ 8.7 Ki 2
LFBIVGMGSSDSAY 8.7 Ki 2
AILQOERCUFVJMB 8.6 Ki 2
WNNZZRWQUYRLFF 8.6 IC50 2
DOIUTSAXPOMBSB 8.6 Ki 2
FOLRUTAUDNCQAE 8.5 IC50 2
VRDBJWJUZBNNGQ 8.5 Ki 2
ULEAFQYUMKDDJU 8.5 Ki 2
HIOYYLSBJMMPNZ 8.5 IC50 2
HKSZLNNOFSGOKW 8.5 Kd 213
KXTWNPILDAXGMS 8.4 Ki 2
WMPRQJNNYNQQIY 8.4 Ki 2
TYBGMAHKOCIODO 8.4 Ki 2
VFPDTTYPIIITKQ 8.4 Ki 2
WZHYYHVLAMIXKN 8.3 IC50 2
XEGXJBWNOCJXQI 8.3 Ki 2
WBYAJDDXRYYJOT 8.2 IC50 2
KQLHECVWPJTIGF 8.2 IC50 2
SDBZHNNKKXPNRV 8.2 Ki 2
KHVXVEAQTZXJAO 8.1 Ki 2
FLEAYYMORDPWAJ 8.1 Ki 90
HKSZLNNOFSGOKW 8.1 IC50 408
NIAZCQPGKHTKAY 8.1 Ki 2
QECHNSUNXZVJGC 8.1 Ki 2
RSBIYYBKMTVJFZ 8.0 Ki 2
GLDSKRNGVVYJAB 8.0 Kd 16
MVJMMLFMPWITEJ 8.0 Ki 110
SGZZQKMOFHIDKW 8.0 Kd 13
FPYJSJDOHRDAMT 8.0 Ki 4
KUYINOAQXYFSBK 8.0 Ki 2
LRZKRKDRHKBUGU 8.0 Ki 2
CEUUNSLVUOVLFP 8.0 Ki 2
IETJKSWTKVOWBN 8.0 Ki 2
DIXMBHMNEHPFCX 7.9 IC50 12
JQSJFFRJYAGFLL 7.9 IC50 2
2D structure