Target Details
| UniProt AC | Q14164 |
|---|---|
| Gene Symbol | IKBKE |
| Protein Name | Inhibitor of nuclear factor kappa-B kinase subunit epsilon |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 596
- Clinical molecules 14
- Avg pChEMBL 7.38
KEGG Pathways (18)
- Alcoholic liver disease
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - receptor activation
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- NOD-like receptor signaling pathway
- RIG-I-like receptor signaling pathway
- Toll-like receptor signaling pathway
Active Molecules (596)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CLYZLUAUBTXCPL
|
6.9 | IC50 | 7 | — | |
DUUHSIDQKSIHGY
|
6.9 | IC50 | 2 | — | |
FXKNBVDEHBSMEE
|
6.9 | IC50 | 2 | — | |
KEZNARMJBJOFQB
|
6.9 | IC50 | 2 | — | |
KPJNILHFVBUXEY
|
6.9 | IC50 | 2 | — | |
OOZSAGRBHKWOLQ
|
6.9 | IC50 | 2 | — | |
YOUNKSLLTJRACV
|
6.9 | IC50 | 2 | — | |
OOMBFNDWQIGHEK
|
6.9 | Kd | 22 | — | |
RWFVTYXPQZEJCN
|
6.9 | IC50 | 3 | — | |
KLUCDSGOLCBPFE
|
6.9 | IC50 | 3 | — | |
OWRXHGAFWZFFCW
|
6.9 | Ki | 113 | — | |
ZGDYBJXDIXVTLV
|
6.9 | Ki | 54 | — | |
PNMCLCQZSVIVDN
|
6.9 | IC50 | 2 | — | |
FQMQKRIYLONZDU
|
6.8 | IC50 | 2 | — | |
GJVSHKMQEGTVTJ
|
6.8 | IC50 | 2 | — | |
RTLYKZQELDVJNY
|
6.8 | IC50 | 2 | — | |
YYPXOMDDWZLVDO
|
6.8 | IC50 | 2 | — | |
DGEFLIVVPLYQKC
|
6.8 | IC50 | 2 | — | |
HTIICNKYFZGUBY
|
6.8 | IC50 | 2 | — | |
UEESRKKBPBMNHE
|
6.8 | IC50 | 2 | — | |
YPWCKOYUDFFQRI
|
6.8 | IC50 | 2 | — | |
XMFSUNMVGUQZBX
|
6.8 | IC50 | 2 | — | |
BMGQWWVMWDBQGC
|
6.8 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.8 | Kd | 91 | Yes | |
LLHGFGUOUWJTLQ
|
6.8 | IC50 | 3 | — | |
PROLIXHVRCJEFH
|
6.8 | Ki | 46 | — | |
QNONXXVGNAZLMI
|
6.8 | IC50 | 2 | — | |
UKBGBACORPRCGG
|
6.8 | IC50 | 17 | — | |
IFIYTVUHPORWKB
|
6.8 | IC50 | 3 | — | |
UOPCRSIUYMGQCP
|
6.8 | IC50 | 6 | — | |
XZXHXSATPCNXJR
|
6.8 | Kd | 165 | Yes | |
XVLUNMSWJVTNRP
|
6.8 | IC50 | 4 | — | |
DKZYXHCYPUVGAF
|
6.7 | Kd | 112 | — | |
WZWSPTDKPFXDGL
|
6.7 | IC50 | 2 | — | |
QYKSYJHYCDJRQT
|
6.7 | IC50 | 2 | — | |
RDFHITQJRDVSMP
|
6.7 | IC50 | 5 | — | |
JNXJKTXDSPWNRP
|
6.7 | Ki | 30 | — | |
JQSSJNGHYKCXQI
|
6.7 | IC50 | 2 | — | |
QSNAYNYUEDJOLU
|
6.7 | IC50 | 2 | — | |
SYMILEXMAHCATG
|
6.7 | IC50 | 2 | — | |
ZGZVRPRSFXRGCF
|
6.7 | Ki | 76 | — | |
ZUDLFDOJAKMMDT
|
6.7 | IC50 | 2 | — | |
ASDFEOAEPCPHHU
|
6.7 | IC50 | 2 | — | |
BTUAQQDZVLCPFW
|
6.7 | IC50 | 2 | — | |
RYGAYBGVUQJRJA
|
6.7 | IC50 | 3 | — | |
ULGOPTXVFIQHMI
|
6.7 | IC50 | 3 | — | |
IZDUBCLXNXGBOL
|
6.7 | IC50 | 2 | — | |
MRXMSGWSWWMSMF
|
6.7 | IC50 | 2 | — | |
RURLEFVQRJFOOD
|
6.7 | IC50 | 2 | — | |
LOLPPWBBNUVNQZ
|
6.7 | Kd | 97 | Yes |