Target Details
| UniProt AC | Q14164 |
|---|---|
| Gene Symbol | IKBKE |
| Protein Name | Inhibitor of nuclear factor kappa-B kinase subunit epsilon |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 596
- Clinical molecules 14
- Avg pChEMBL 7.38
KEGG Pathways (18)
- Alcoholic liver disease
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - receptor activation
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- NOD-like receptor signaling pathway
- RIG-I-like receptor signaling pathway
- Toll-like receptor signaling pathway
Active Molecules (596)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VCFDMLBPASGZTP
|
7.2 | Ki | 38 | — | |
BGXAJMOKNLNIKN
|
7.2 | IC50 | 2 | — | |
HYKUTXSZGOOHPE
|
7.2 | IC50 | 2 | — | |
YJYNURQSPOYQLL
|
7.2 | IC50 | 2 | — | |
SQZVSGZHYGZMTP
|
7.2 | IC50 | 2 | — | |
NHSSQLZJTUWHPU
|
7.2 | IC50 | 2 | — | |
FQMLNDAGKXRMPL
|
7.2 | IC50 | 2 | — | |
VOYZWDQJVPQGCO
|
7.2 | IC50 | 9 | — | |
ZRQQVUBJGLMDQR
|
7.2 | IC50 | 2 | — | |
IQRLNHJUFLQKGU
|
7.1 | IC50 | 2 | — | |
JUWVGQDRIAVTIK
|
7.1 | IC50 | 3 | — | |
ZCCPLJOKGAACRT
|
7.1 | Kd | 599 | — | |
CGFPGAHHLFCHCL
|
7.1 | IC50 | 2 | — | |
XXSJUYSLBGBRGF
|
7.1 | IC50 | 2 | — | |
BYGZCGOGQACGKA
|
7.1 | IC50 | 2 | — | |
LPISIKGCJPHMTC
|
7.1 | IC50 | 2 | — | |
ALNFAQPPDFVBLE
|
7.1 | IC50 | 2 | — | |
UDLCUPNAFTWKLG
|
7.1 | IC50 | 2 | — | |
CIBIQJXLLSSQGJ
|
7.1 | IC50 | 2 | — | |
VLQLXNFFVREKBK
|
7.1 | IC50 | 3 | — | |
DYVYNFDWCPVADF
|
7.1 | IC50 | 2 | — | |
PNYUSFRZJAPJCP
|
7.1 | IC50 | 2 | — | |
XHGRACBJXGTCJY
|
7.1 | IC50 | 2 | — | |
NDSBUHYDEKJESH
|
7.0 | IC50 | 2 | — | |
UDQFLASTRAMKLW
|
7.0 | IC50 | 3 | — | |
HPYDIJUSTZXNRN
|
7.0 | IC50 | 2 | — | |
JOPQBRQUFRAGQH
|
7.0 | IC50 | 2 | — | |
ANVBJUPKQASFMW
|
7.0 | IC50 | 3 | — | |
VJMPKACKJOXZGT
|
7.0 | IC50 | 2 | — | |
VWWBXTRZUJUTHA
|
7.0 | IC50 | 2 | — | |
OUTINXWZDNJANR
|
7.0 | IC50 | 2 | — | |
QTSKVQLIRGIGDV
|
7.0 | IC50 | 3 | — | |
MJTMCXPFKSSYRZ
|
7.0 | IC50 | 2 | — | |
VNDWQCSOSCCWIP
|
7.0 | Ki | 39 | Yes | |
XAJOPTJESFDNGL
|
7.0 | IC50 | 2 | — | |
YOFJPZPGHXWQJB
|
7.0 | IC50 | 5 | — | |
IHPBCWXBUXLKAX
|
7.0 | IC50 | 2 | — | |
QKAVQJBBCRMGMX
|
7.0 | IC50 | 3 | — | |
BTIIUKSFWMYFNV
|
7.0 | IC50 | 6 | — | |
ISADMOXHYKRVEW
|
7.0 | IC50 | 2 | — | |
SPYTVKZEORYOEZ
|
7.0 | IC50 | 2 | — | |
SSAUMSLDIATKRC
|
7.0 | IC50 | 3 | — | |
UYIHWPCEDZKSLA
|
7.0 | IC50 | 2 | — | |
IXANCEFCAMWOSC
|
7.0 | IC50 | 2 | — | |
SINJOIVMLYFADD
|
7.0 | IC50 | 5 | — | |
AZBYFLYSUMYTKS
|
6.9 | IC50 | 2 | — | |
BKJRFMUYVNJZKE
|
6.9 | IC50 | 2 | — | |
GFHRPONHRZBFNC
|
6.9 | IC50 | 3 | — | |
PDMRUTWXKCFDFD
|
6.9 | IC50 | 2 | — | |
CGELHDCKISPXTF
|
6.9 | IC50 | 2 | — |