Target Details
| UniProt AC | Q14164 |
|---|---|
| Gene Symbol | IKBKE |
| Protein Name | Inhibitor of nuclear factor kappa-B kinase subunit epsilon |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 596
- Clinical molecules 14
- Avg pChEMBL 7.38
KEGG Pathways (18)
- Alcoholic liver disease
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - receptor activation
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- NOD-like receptor signaling pathway
- RIG-I-like receptor signaling pathway
- Toll-like receptor signaling pathway
Active Molecules (596)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OWTXNTZZHGTTPX
|
7.6 | IC50 | 2 | — | |
VKBFHTIUXUCYRQ
|
7.6 | Ki | 66 | — | |
WPHKIQPVPYJNAX
|
7.6 | Ki | 81 | — | |
WSZQEIWUWGBMDJ
|
7.6 | IC50 | 2 | — | |
YDRISZZAAFDOPR
|
7.6 | IC50 | 2 | — | |
YVRJIQLODAYFSS
|
7.6 | IC50 | 2 | — | |
YZWVXQXPLIUUGA
|
7.6 | IC50 | 2 | — | |
MBYYLRDCKQHUGM
|
7.6 | IC50 | 3 | — | |
HNDZOIQVTDQHDZ
|
7.6 | IC50 | 2 | — | |
WEFRCKPVMWDRAK
|
7.5 | IC50 | 5 | — | |
KPELCBIAAJVUQI
|
7.5 | IC50 | 3 | — | |
LUIAXPRIBAAQLN
|
7.5 | IC50 | 2 | — | |
IWILCSQODDAQDC
|
7.5 | IC50 | 2 | — | |
OAYVEVAGVZYBHT
|
7.5 | IC50 | 2 | — | |
XEHKYAPSLVQNOG
|
7.5 | IC50 | 2 | — | |
LIYOMPYVPWOZJX
|
7.5 | IC50 | 2 | — | |
YTKXJIKRZSXVIP
|
7.5 | IC50 | 2 | — | |
AUVLVGAPOCTIAE
|
7.5 | IC50 | 3 | — | |
CAVHGBLDRHUXIQ
|
7.5 | IC50 | 3 | — | |
GBDGRXDOLFLBAV
|
7.5 | IC50 | 3 | — | |
GDMLXKZMNHJKNI
|
7.5 | IC50 | 3 | — | |
GHZHOTWEULSCJL
|
7.5 | IC50 | 3 | — | |
GJAQYJWEEXUKPK
|
7.5 | IC50 | 3 | — | |
IAQRFOBNZQJZEU
|
7.5 | IC50 | 3 | — | |
IFNASLLOEPLWNG
|
7.5 | IC50 | 3 | — | |
IHWPMUHWLMAGRM
|
7.5 | IC50 | 3 | — | |
IQQCLKRZDHVEJC
|
7.5 | IC50 | 3 | — | |
KNCDEVRJJHZTFP
|
7.5 | IC50 | 3 | — | |
LRDQYJRVAAGHEK
|
7.5 | IC50 | 3 | — | |
MAGYPARKFHXVPO
|
7.5 | IC50 | 3 | — | |
MGUWFXNRNXEUEB
|
7.5 | IC50 | 3 | — | |
NMJIAJITODSLIF
|
7.5 | IC50 | 3 | — | |
OYQSRSUSXBDIKK
|
7.5 | IC50 | 3 | — | |
OYQSRSUSXBDIKK
|
7.5 | IC50 | 3 | — | |
PRELXQNFYRQFTQ
|
7.5 | IC50 | 3 | — | |
QPWPSCNQQGTOFW
|
7.5 | IC50 | 3 | — | |
QYECLBIGLCTRAG
|
7.5 | IC50 | 3 | — | |
SDJZXXAGAUAGTD
|
7.5 | IC50 | 3 | — | |
VHGHPWKEDSVCPO
|
7.5 | IC50 | 3 | — | |
WUOSUEXRIIWVRA
|
7.5 | IC50 | 3 | — | |
XFQGLEVRHJHNBR
|
7.5 | IC50 | 3 | — | |
XWAAZPHGKVWIBO
|
7.5 | IC50 | 3 | — | |
XYLDHWOGWNKCSD
|
7.5 | IC50 | 3 | — | |
YLNRUJJGFNIFJI
|
7.5 | IC50 | 3 | — | |
ZTDINRKSUABPHP
|
7.5 | IC50 | 3 | — | |
LARUOSVANYWRFG
|
7.5 | IC50 | 2 | — | |
LBFKDBMDAOTADZ
|
7.5 | IC50 | 3 | — | |
WTRFGRRHMCNXPV
|
7.5 | IC50 | 2 | — | |
AKBNGGYXMZTHEB
|
7.5 | IC50 | 5 | — | |
CYCDEYIKBNVSHA
|
7.5 | IC50 | 2 | — |