Target Details
| UniProt AC | Q14164 |
|---|---|
| Gene Symbol | IKBKE |
| Protein Name | Inhibitor of nuclear factor kappa-B kinase subunit epsilon |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 596
- Clinical molecules 14
- Avg pChEMBL 7.38
KEGG Pathways (18)
- Alcoholic liver disease
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - receptor activation
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- NOD-like receptor signaling pathway
- RIG-I-like receptor signaling pathway
- Toll-like receptor signaling pathway
Active Molecules (596)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OTDPQDOEHSIHCV
|
8.1 | IC50 | 2 | — | |
YFBHNTGOTRHQLM
|
8.1 | IC50 | 3 | — | |
ZNTAAWCMFQAOKC
|
8.1 | IC50 | 3 | — | |
LZVZBSNKTPVPEB
|
8.0 | IC50 | 2 | — | |
IITKALICJDNWMU
|
8.0 | IC50 | 2 | — | |
ZCTTVOCGTHIYCW
|
8.0 | IC50 | 2 | — | |
AAEIQQDLGQELDQ
|
8.0 | IC50 | 2 | — | |
BPNSGZHWOGXFQP
|
8.0 | IC50 | 3 | — | |
JNYUZMNVAQNKRU
|
8.0 | IC50 | 2 | — | |
KHKGVBAGOBQZSK
|
8.0 | IC50 | 2 | — | |
MZKFOXRCMQMVAM
|
8.0 | IC50 | 3 | — | |
NQVRHDTYGKEBDT
|
8.0 | IC50 | 2 | — | |
QNAQWEYXUVCFQZ
|
8.0 | IC50 | 3 | — | |
XBFXJAXJSWLRPR
|
8.0 | IC50 | 2 | — | |
XJXPKTHMXWGQPH
|
8.0 | IC50 | 5 | — | |
ZXXUISVZQNQVSN
|
8.0 | IC50 | 2 | — | |
UBBGWCKRFYZCTO
|
8.0 | IC50 | 2 | — | |
WPWPOCITVIKSCW
|
8.0 | IC50 | 2 | — | |
FTVIWWJJRCVHSZ
|
8.0 | IC50 | 2 | — | |
HKVLGLZTELKITJ
|
8.0 | IC50 | 2 | — | |
IVNHCMJOZZBIAP
|
8.0 | IC50 | 2 | — | |
FNVPRBKVDPEQJB
|
8.0 | IC50 | 3 | — | |
OOYRAPOOQHGEBB
|
8.0 | IC50 | 3 | — | |
RVVXQNJZYNFBHM
|
8.0 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
8.0 | Kd | 289 | Yes | |
VZSXBDWSTNVNJE
|
8.0 | IC50 | 2 | — | |
IYLJIJFVSGZAIK
|
8.0 | IC50 | 2 | — | |
MZHPEELZCYWEHG
|
8.0 | IC50 | 6 | — | |
RSUQGUXLJAJYCT
|
7.9 | IC50 | 2 | — | |
TUIAFUOZECMRAZ
|
7.9 | IC50 | 2 | — | |
URHODGROVLUHQW
|
7.9 | IC50 | 3 | — | |
MZUYZYAQDFGDQX
|
7.9 | IC50 | 2 | — | |
RNJBPIVRBMZSMD
|
7.9 | IC50 | 2 | — | |
UAROTPQRUDFOGH
|
7.9 | IC50 | 2 | — | |
WSBKHPYKYJZQTB
|
7.9 | IC50 | 2 | — | |
BJJXTIWXVHNEJL
|
7.9 | IC50 | 2 | — | |
IOIONYMZILVMCR
|
7.9 | IC50 | 2 | — | |
AXFMFRVMFJMHRE
|
7.9 | IC50 | 2 | — | |
AYUVNFPAFJUWQW
|
7.8 | IC50 | 2 | — | |
GHMJUVTUHKPGKE
|
7.8 | IC50 | 3 | — | |
HPLAJCJEPOOJCG
|
7.8 | IC50 | 3 | — | |
MCVZGUNLGAFYGU
|
7.8 | IC50 | 2 | — | |
MSXLIUGGWDIIKN
|
7.8 | IC50 | 3 | — | |
XKQXMMZJRYXZOV
|
7.8 | IC50 | 3 | — | |
YIBZCPJGTIQSGV
|
7.8 | IC50 | 2 | — | |
BDDBUOVVYOJPSW
|
7.8 | IC50 | 2 | — | |
CGDQNIWGTMYVJH
|
7.8 | IC50 | 2 | — | |
PPLYZIXDSCRZFR
|
7.8 | IC50 | 2 | — | |
FONLVAFSTIESFR
|
7.8 | IC50 | 2 | — | |
PQVPIJFBUFHXCN
|
7.8 | IC50 | 2 | — |