Target Details
| UniProt AC | Q14164 |
|---|---|
| Gene Symbol | IKBKE |
| Protein Name | Inhibitor of nuclear factor kappa-B kinase subunit epsilon |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 596
- Clinical molecules 14
- Avg pChEMBL 7.38
KEGG Pathways (18)
- Alcoholic liver disease
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - receptor activation
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- NOD-like receptor signaling pathway
- RIG-I-like receptor signaling pathway
- Toll-like receptor signaling pathway
Active Molecules (596)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CTNPALGJUAXMMC
|
6.3 | Kd | 151 | — | |
GLXBQRZXUMNQRW
|
6.3 | IC50 | 2 | — | |
PIQCTGMSNWUMAF
|
6.3 | Kd | 137 | Yes | |
VSGIYMAWHNSRDN
|
6.3 | IC50 | 2 | — | |
KOZFSFOOLUUIGY
|
6.3 | Kd | 88 | Yes | |
CBFGRAMTCIRLOX
|
6.3 | Ki | 3 | — | |
KTEIFNKAUNYNJU
|
6.3 | Ki | 48 | — | |
SMAIRFQFHKTXBK
|
6.3 | IC50 | 2 | — | |
MERPPDGMBNDZGS
|
6.3 | IC50 | 2 | — | |
RWJIWEQYLOKEBO
|
6.3 | IC50 | 2 | — | |
BRHAIUXYHUZNFP
|
6.3 | IC50 | 2 | — | |
IMXLNRXFUOHHDN
|
6.3 | IC50 | 2 | — | |
PBCZSGKMGDDXIJ
|
6.3 | Kd | 68 | Yes | |
ZTLALBZROUPCEA
|
6.3 | IC50 | 2 | — | |
BWZFHPDMLLCYGG
|
6.3 | IC50 | 2 | — | |
CYSDRDWNFDQHMX
|
6.3 | IC50 | 2 | — | |
JJEHKOXQJFSVQK
|
6.3 | IC50 | 2 | — | |
NSNZIHNPWOUVQN
|
6.3 | IC50 | 2 | — | |
AGRUJTXFZAUTCB
|
6.3 | IC50 | 2 | — | |
BMPKLAIDXFLOJP
|
6.3 | IC50 | 2 | — | |
CFBXWHPXNROFFK
|
6.3 | IC50 | 4 | — | |
CYKQBRKJEQQTHD
|
6.3 | IC50 | 2 | — | |
HDPFOBSEWXADBZ
|
6.3 | IC50 | 2 | — | |
HSTCZBIJGXTJBW
|
6.3 | IC50 | 2 | — | |
MBMXQMPCISCAST
|
6.3 | IC50 | 2 | — | |
NGRIQWBQAPFNJW
|
6.3 | IC50 | 2 | — | |
RHAHFLIAPLIWKN
|
6.3 | IC50 | 2 | — | |
ZQAHHQOAUDLNLW
|
6.3 | IC50 | 2 | — | |
FJJRVGSILLVPKU
|
6.2 | IC50 | 2 | — | |
CIKDZQBTQZZADZ
|
6.2 | IC50 | 3 | — | |
ZVBIBRJWIINCLT
|
6.2 | IC50 | 2 | — | |
SYMILEXMAHCATG
|
6.2 | IC50 | 2 | — | |
ZNBXHMDTLSAOFO
|
6.2 | IC50 | 2 | — | |
BHMSKCZYCFPYKC
|
6.2 | IC50 | 2 | — | |
XXDNMKSTCJGGQP
|
6.2 | IC50 | 2 | — | |
PMEYAHBGTDHJEZ
|
6.2 | IC50 | 2 | — | |
WINHZLLDWRZWRT
|
6.2 | Kd | 201 | Yes | |
ADLPKFFMGIJZIM
|
6.2 | Ki | 44 | — | |
BLQYVHBZHAISJM
|
6.2 | Ki | 54 | — | |
FUIFXIHDSHGQPX
|
6.2 | IC50 | 2 | — | |
JJGSOVIZOMZMCS
|
6.2 | Ki | 35 | — | |
KUNZDWIFPOMUOX
|
6.2 | Ki | 36 | — | |
RTYJMUXLFRYRBU
|
6.2 | Ki | 35 | — | |
SGSXSDRBQOSVBH
|
6.2 | IC50 | 2 | — | |
UQNNJYLAPYGZBD
|
6.2 | Ki | 28 | — | |
GIWAUMWDROOOBY
|
6.2 | IC50 | 2 | — | |
AYCPARAPKDAOEN
|
6.2 | Kd | 73 | — | |
CMRSPQFHPQBQIK
|
6.2 | IC50 | 2 | — | |
RMTFITAOVDYEPI
|
6.2 | IC50 | 2 | — | |
OYONTEXKYJZFHA
|
6.2 | Kd | 69 | Yes |