Target Details
| UniProt AC | Q14164 |
|---|---|
| Gene Symbol | IKBKE |
| Protein Name | Inhibitor of nuclear factor kappa-B kinase subunit epsilon |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 596
- Clinical molecules 14
- Avg pChEMBL 7.38
KEGG Pathways (18)
- Alcoholic liver disease
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - receptor activation
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- NOD-like receptor signaling pathway
- RIG-I-like receptor signaling pathway
- Toll-like receptor signaling pathway
Active Molecules (596)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MHPBLCYPFBBOND
|
6.7 | IC50 | 6 | — | |
PEGMEQCMRMUMBG
|
6.7 | IC50 | 2 | — | |
NLPNLVFDNONUOB
|
6.6 | IC50 | 2 | — | |
ZIRAJQJDABKSFH
|
6.6 | IC50 | 2 | — | |
GJOXRIYWDHESDF
|
6.6 | Ki | 27 | — | |
PYVMYBZZIWFCPE
|
6.6 | IC50 | 2 | — | |
BGAUWQRNGCAKTK
|
6.6 | IC50 | 2 | — | |
AFZREGWWRXQGGC
|
6.6 | IC50 | 2 | — | |
OGCZIWWQVLKYDK
|
6.6 | IC50 | 2 | — | |
WOTWXKACTZFRQE
|
6.6 | IC50 | 4 | — | |
KZXWFUQZOSWUCY
|
6.6 | IC50 | 2 | — | |
KMIUIHAGKAMAMN
|
6.6 | IC50 | 2 | — | |
ZEEVDVUFURMNEH
|
6.6 | IC50 | 2 | — | |
GANHRJNVDOQXBZ
|
6.5 | IC50 | 2 | — | |
RFYVLIYJZUYOAT
|
6.5 | IC50 | 2 | — | |
SLEWGGZPOQNVSU
|
6.5 | Kd | 22 | — | |
CPOMPMCLFHSOKH
|
6.5 | IC50 | 2 | — | |
IUSHILFEMDZEFI
|
6.5 | IC50 | 2 | — | |
OMSMAWMALYCJCB
|
6.5 | IC50 | 2 | — | |
QDJHWYVWXZCCGP
|
6.5 | IC50 | 2 | — | |
UDNWHJPQDRSGDI
|
6.5 | IC50 | 2 | — | |
IUYVWTVARMTLCH
|
6.5 | IC50 | 2 | — | |
PMXKKMZIBVSKTC
|
6.5 | IC50 | 2 | — | |
VWJJCQKYLQGLKH
|
6.5 | IC50 | 2 | — | |
ZZSBPGIGIUFJRA
|
6.5 | Kd | 46 | — | |
OESXQVFTYMQBFH
|
6.5 | IC50 | 2 | — | |
SSAAGCQGRIMQSH
|
6.5 | IC50 | 2 | — | |
YXNUVQPEHUKSLS
|
6.5 | IC50 | 2 | — | |
CLVOFVSKXGTJMX
|
6.5 | IC50 | 2 | — | |
NHEUUFMAYLMPKA
|
6.5 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
6.5 | Kd | 191 | — | |
JOOXLOJCABQBSG
|
6.4 | Kd | 139 | — | |
HDOTZQLJXWSXIO
|
6.4 | IC50 | 2 | — | |
DWBFATQGRAYQFC
|
6.4 | IC50 | 2 | — | |
UANVBHMEXMGHSB
|
6.4 | IC50 | 2 | — | |
WXNQCJRSDVNYKO
|
6.4 | IC50 | 2 | — | |
YSJYNAPMKLZIGV
|
6.4 | IC50 | 2 | — | |
GJKVMXDBPDDFHI
|
6.4 | Ki | 27 | — | |
MHWHPWMWKYXCRJ
|
6.4 | Ki | 32 | — | |
NKTGILZAOLEZPR
|
6.4 | IC50 | 2 | — | |
VSVWQTDDGQSGHP
|
6.4 | Ki | 51 | — | |
FLBNLJLONKAPLR
|
6.4 | Kd | 31 | — | |
DCRFLNHKMKYMQP
|
6.4 | IC50 | 2 | — | |
MJBVMFNLYNJFSW
|
6.4 | IC50 | 2 | — | |
NBXRQAXVXWKQJZ
|
6.4 | IC50 | 2 | — | |
NZELJWLQMFWZDX
|
6.4 | IC50 | 2 | — | |
LSYVMTFICMPMTL
|
6.4 | IC50 | 2 | — | |
BXMGOFSMDOETKZ
|
6.3 | IC50 | 2 | — | |
UOFZOMWGIVJIKW
|
6.3 | IC50 | 3 | — | |
WWRBLGBEFCCCCB
|
6.3 | IC50 | 2 | — |