Target Details
| UniProt AC | Q14164 |
|---|---|
| Gene Symbol | IKBKE |
| Protein Name | Inhibitor of nuclear factor kappa-B kinase subunit epsilon |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 596
- Clinical molecules 14
- Avg pChEMBL 7.38
KEGG Pathways (18)
- Alcoholic liver disease
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - receptor activation
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- NOD-like receptor signaling pathway
- RIG-I-like receptor signaling pathway
- Toll-like receptor signaling pathway
Active Molecules (596)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.4 | IC50 | 408 | — | |
HVZSQXWYDLQJTQ
|
9.3 | IC50 | 2 | — | |
LNIVPTBCCJSTCB
|
9.2 | IC50 | 2 | — | |
RGVXQILQOSLWGS
|
9.2 | IC50 | 2 | — | |
BXLOFFCDXFSKIE
|
9.1 | IC50 | 2 | — | |
GVXJFRXNNLRSLI
|
9.1 | IC50 | 2 | — | |
LYMQARVHTYDQHO
|
9.0 | IC50 | 2 | — | |
RXRLWNRSQUSJOR
|
8.9 | IC50 | 2 | — | |
HSLJCXAGEGDBAU
|
8.9 | IC50 | 2 | — | |
RQMSNFNMLUFOPR
|
8.8 | IC50 | 2 | — | |
PRBYIDLQEMMFNC
|
8.8 | IC50 | 2 | — | |
JHCYMEMCUXVAIR
|
8.8 | IC50 | 2 | — | |
UNZLCMSGBFLOLV
|
8.7 | IC50 | 2 | — | |
VIURSDPOFRRBCH
|
8.7 | IC50 | 2 | — | |
ZULNHRNAEOVNJO
|
8.7 | IC50 | 2 | — | |
DYRXRIMUJAAMQI
|
8.7 | IC50 | 2 | — | |
ABJMUSKMRCDMPE
|
8.7 | IC50 | 3 | — | |
AEPJRUANSIXNRU
|
8.7 | IC50 | 3 | — | |
BCPZVZDYGYPCDP
|
8.7 | IC50 | 3 | — | |
CGORDIYPCGPLIZ
|
8.7 | IC50 | 3 | — | |
CYSNREWCZKAVDY
|
8.7 | IC50 | 3 | — | |
DFQJNFGZAMXNJM
|
8.7 | IC50 | 3 | — | |
GHZHOTWEULSCJL
|
8.7 | IC50 | 3 | — | |
GRPKFQBLNWZZJC
|
8.7 | IC50 | 3 | — | |
GXCCDZRRVFNQMR
|
8.7 | IC50 | 3 | — | |
HZRJHVDNTDBTOZ
|
8.7 | IC50 | 8 | — | |
ICTZCEFKLIZUFV
|
8.7 | IC50 | 3 | — | |
JOMSKNSFOAKBRO
|
8.7 | IC50 | 3 | — | |
JSWSNMUJSFRFCL
|
8.7 | IC50 | 3 | — | |
KAKYKHXANDESRF
|
8.7 | IC50 | 3 | — | |
KOLYMXQYZQEXIF
|
8.7 | IC50 | 3 | — | |
OCMXFNGLZPKTFI
|
8.7 | IC50 | 3 | — | |
PMQODLVRCODLJS
|
8.7 | IC50 | 3 | — | |
QRQGHALETIKFSZ
|
8.7 | IC50 | 3 | — | |
QUOKNSGMLFDHHY
|
8.7 | IC50 | 3 | — | |
VILUZAYZRGMLRF
|
8.7 | IC50 | 3 | — | |
WNPBFIJEFIXYRM
|
8.7 | IC50 | 3 | — | |
WRMHBKKOYNOLHH
|
8.7 | IC50 | 2 | — | |
XCYPLUKAXOGVDS
|
8.7 | IC50 | 3 | — | |
YPUJLPFDSVVFMZ
|
8.7 | IC50 | 3 | — | |
YRMKHJKXKFHXMK
|
8.7 | IC50 | 3 | — | |
ZUUSJSDRSNEYLL
|
8.7 | IC50 | 3 | — | |
QRICOSSIVLKBBT
|
8.7 | IC50 | 2 | — | |
LDJRWCYJKDXGCY
|
8.6 | IC50 | 2 | — | |
SSFXUEWPQPILFO
|
8.6 | IC50 | 2 | — | |
WQFRKFJYPSEBPY
|
8.6 | IC50 | 2 | — | |
HXAYGARTNPQTPX
|
8.6 | IC50 | 2 | — | |
XZIIRCPKAFVFHW
|
8.6 | IC50 | 2 | — | |
XSGVWMDUOODJTB
|
8.6 | IC50 | 2 | — | |
XKXKAOTUKINWLC
|
8.5 | IC50 | 2 | — |