Target Details
| UniProt AC | Q14145 |
|---|---|
| Gene Symbol | KEAP1 |
| Protein Name | Kelch-like ECH-associated protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07707 (BACK) PF00651 (BTB) PF01344 (Kelch_1) PF24681 (Kelch_KLHDC2_KLHL20_DRC7) |
Summary
- Multi-target molecules 558
- Clinical molecules 0
- Avg pChEMBL 7.21
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (558)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YVVSLYWCORNKAO
|
7.3 | IC50 | 2 | — | |
YYIAYPKFORFCIY
|
7.3 | IC50 | 2 | — | |
YZJHIJHDIPVFFH
|
7.3 | IC50 | 2 | — | |
ZDNGJXBUEQNFBQ
|
7.3 | IC50 | 2 | — | |
ZEXIQZWCZZOHLR
|
7.3 | IC50 | 2 | — | |
ZHDBZJLNJLJQMN
|
7.3 | IC50 | 2 | — | |
ZKSQTPIKIPUMJG
|
7.3 | IC50 | 2 | — | |
ZSYJPILCQQZFGC
|
7.3 | IC50 | 2 | — | |
ZXWYNATUZLXLKZ
|
7.3 | IC50 | 2 | — | |
PWKJRVHFVZDUJL
|
7.2 | Kd | 2 | — | |
AHNXOLRIYAUDAJ
|
7.2 | Kd | 2 | — | |
ILYPAKWDDIPWBD
|
7.2 | IC50 | 2 | — | |
IMRNAESQPBZZKY
|
7.2 | Kd | 2 | — | |
CHFWRHMYWKNWOD
|
7.2 | Kd | 2 | — | |
JAVOONPTJYTDCV
|
7.2 | IC50 | 2 | — | |
BVWKAUMFAYUKCN
|
7.2 | IC50 | 2 | — | |
SDNGUWKKARNBMG
|
7.2 | IC50 | 2 | — | |
YNVNINGXKVYVIH
|
7.2 | IC50 | 2 | — | |
UVJKKKIWFDQRIO
|
7.1 | IC50 | 2 | — | |
BPXRLRWCXHOGKW
|
7.1 | IC50 | 2 | — | |
UQMFOGQVOSBRDN
|
7.1 | IC50 | 2 | — | |
FCUHBMJCDSGVHP
|
7.1 | Kd | 2 | — | |
ZHCPWSXUYVGNBT
|
7.1 | Ki | 2 | — | |
BYDRCKDNJKPUKF
|
7.1 | IC50 | 2 | — | |
IRTRBIIUERHWMH
|
7.1 | IC50 | 2 | — | |
FEYLEFUBCXEKAO
|
7.1 | IC50 | 2 | — | |
NFGAQVYFVVMRES
|
7.1 | IC50 | 2 | — | |
XIOLQNIMTYKYJQ
|
7.0 | IC50 | 2 | — | |
ASUYATVKGAAOID
|
7.0 | IC50 | 2 | — | |
RRPUEYFUGJMNBJ
|
7.0 | IC50 | 2 | — | |
CDAORYDEXZVXAW
|
7.0 | IC50 | 2 | — | |
DDOCYQXGLAMLTA
|
7.0 | IC50 | 2 | — | |
ZLGGCMKZTJOJRY
|
7.0 | Ki | 2 | — | |
RWWBWFNNADGJJB
|
7.0 | IC50 | 2 | — | |
QWRFZAZSUNMQDD
|
7.0 | Kd | 2 | — | |
OLNOWMNEHRFYCP
|
7.0 | Kd | 2 | — | |
NVQFDGYHTTZFJR
|
7.0 | IC50 | 2 | — | |
PWKJRVHFVZDUJL
|
7.0 | Kd | 2 | — | |
JNGVVGXJVLYMRP
|
6.9 | IC50 | 2 | — | |
ONBIYOXDYQDZBR
|
6.9 | IC50 | 2 | — | |
POXZWUFGBAMZNF
|
6.9 | IC50 | 2 | — | |
SEYURAKXESNAMM
|
6.9 | Kd | 2 | — | |
XTOTXBIQVUFPGY
|
6.9 | IC50 | 2 | — | |
ZICYTEWSORSQPC
|
6.9 | IC50 | 2 | — | |
YEVIWEXNDKLEQN
|
6.9 | IC50 | 2 | — | |
IWAWWUSRLVMCRW
|
6.9 | Ki | 2 | — | |
MQNFGUOKPYSZBX
|
6.9 | IC50 | 2 | — | |
RPNAHZQRARAOJE
|
6.9 | IC50 | 2 | — | |
UIPYFTOJSADVTQ
|
6.9 | IC50 | 2 | — | |
BVYWIQHJXAEJOD
|
6.8 | IC50 | 2 | — |