Target Details
| UniProt AC | Q14145 |
|---|---|
| Gene Symbol | KEAP1 |
| Protein Name | Kelch-like ECH-associated protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07707 (BACK) PF00651 (BTB) PF01344 (Kelch_1) PF24681 (Kelch_KLHDC2_KLHL20_DRC7) |
Summary
- Multi-target molecules 558
- Clinical molecules 0
- Avg pChEMBL 7.21
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (558)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HSPMCXSTLBKXFP
|
7.3 | IC50 | 2 | — | |
HSZYGMSIEGUWCB
|
7.3 | IC50 | 2 | — | |
HYGIVHHILZAXKU
|
7.3 | IC50 | 2 | — | |
HZDUCHHJWUKSCD
|
7.3 | IC50 | 2 | — | |
IARGPHHSZQXOSH
|
7.3 | IC50 | 2 | — | |
IDANVQJFZXIQGM
|
7.3 | IC50 | 2 | — | |
IDWGQXZQNPNHGS
|
7.3 | IC50 | 2 | — | |
IGSXVTNHKWFQHY
|
7.3 | IC50 | 2 | — | |
IMPTVJDGGVRIHR
|
7.3 | IC50 | 2 | — | |
IMVRDTIUXGSVRZ
|
7.3 | IC50 | 2 | — | |
IOXXTPJNZJWFCO
|
7.3 | IC50 | 2 | — | |
IPCDQJRZKHHXLK
|
7.3 | IC50 | 2 | — | |
JBWZTQKHRVJEFM
|
7.3 | IC50 | 2 | — | |
JBXYFQNBDRELKW
|
7.3 | IC50 | 2 | — | |
JERKNUJOWYNDMT
|
7.3 | IC50 | 2 | — | |
JHJVCRPWCAVTKW
|
7.3 | IC50 | 2 | — | |
JIZILTYHXGMOFC
|
7.3 | IC50 | 2 | — | |
JJZPWGQPPUTFLQ
|
7.3 | IC50 | 2 | — | |
JKDFOYSIKNRLTR
|
7.3 | IC50 | 2 | — | |
JSKSTRUXUJHPPP
|
7.3 | IC50 | 2 | — | |
JXCOERQLGLXVIK
|
7.3 | IC50 | 2 | — | |
JXCOERQLGLXVIK
|
7.3 | IC50 | 2 | — | |
KEWXNRYLPLVBKW
|
7.3 | IC50 | 2 | — | |
KHKRJIKQDOFQIX
|
7.3 | IC50 | 2 | — | |
KJTROJDEHGPKAA
|
7.3 | IC50 | 2 | — | |
KWDUEIBJQOEQJN
|
7.3 | IC50 | 2 | — | |
KWYMBFUQBRMBQX
|
7.3 | IC50 | 2 | — | |
KZOPELYEZBBUIV
|
7.3 | IC50 | 2 | — | |
LJYJNPDCJALUPO
|
7.3 | IC50 | 2 | — | |
LPMRCDNUPGZGDF
|
7.3 | IC50 | 2 | — | |
MBIUESTWBZOSJW
|
7.3 | IC50 | 2 | — | |
MGIAJNGRXJICFA
|
7.3 | IC50 | 2 | — | |
MMIORKVIDQHGLK
|
7.3 | IC50 | 2 | — | |
MVHXCKOOPXKCMR
|
7.3 | IC50 | 2 | — | |
NLWYXGJADHXGKC
|
7.3 | IC50 | 2 | — | |
NMVOOHUGPIZJBG
|
7.3 | IC50 | 2 | — | |
NVMUELBMBSCZMG
|
7.3 | IC50 | 2 | — | |
NZGGZISVMMEMJX
|
7.3 | IC50 | 2 | — | |
NZGGZISVMMEMJX
|
7.3 | IC50 | 2 | — | |
NZSNWLRCXPWOBC
|
7.3 | IC50 | 2 | — | |
OCRPAIWDRJKOTN
|
7.3 | IC50 | 2 | — | |
OFFIZNQRXWXRFR
|
7.3 | IC50 | 2 | — | |
OLHWMXBKPFRTNX
|
7.3 | IC50 | 2 | — | |
ORCXIWDDBGRHOT
|
7.3 | IC50 | 2 | — | |
PPMXGPZSQLHUHK
|
7.3 | IC50 | 2 | — | |
PPNGGDOOVBFKCD
|
7.3 | IC50 | 2 | — | |
PSAYWSGFKCURFC
|
7.3 | IC50 | 2 | — | |
PSAYWSGFKCURFC
|
7.3 | IC50 | 2 | — | |
QLPRJBMOBGFKTF
|
7.3 | IC50 | 2 | — | |
QRYZXQWLCHRQQQ
|
7.3 | IC50 | 2 | — |