Target Details
| UniProt AC | Q14145 |
|---|---|
| Gene Symbol | KEAP1 |
| Protein Name | Kelch-like ECH-associated protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07707 (BACK) PF00651 (BTB) PF01344 (Kelch_1) PF24681 (Kelch_KLHDC2_KLHL20_DRC7) |
Summary
- Multi-target molecules 558
- Clinical molecules 0
- Avg pChEMBL 7.21
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (558)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BOEKOLYWXVRUED
|
7.3 | IC50 | 2 | — | |
BQKAFUSUOCKJSO
|
7.3 | IC50 | 2 | — | |
BQUWAECBQDXVJF
|
7.3 | IC50 | 2 | — | |
BYWWNBFIESJIJW
|
7.3 | IC50 | 2 | — | |
CEYWUMVWUJLPTE
|
7.3 | IC50 | 2 | — | |
CGULIBNLQTVXJS
|
7.3 | IC50 | 2 | — | |
CHDWDCOIXZPZNY
|
7.3 | IC50 | 2 | — | |
CJTSGSQAUXSAER
|
7.3 | IC50 | 2 | — | |
CPMDCWKBUNBNCQ
|
7.3 | IC50 | 2 | — | |
CQOQRYVBFZKAPT
|
7.3 | IC50 | 2 | — | |
CQYMHLFEMQKUBC
|
7.3 | IC50 | 2 | — | |
CYAWSFDLOYOCFO
|
7.3 | IC50 | 2 | — | |
CYOBABBSHLGCGY
|
7.3 | IC50 | 2 | — | |
CYYQUZIQAPCJLW
|
7.3 | IC50 | 2 | — | |
DHXVRUGBGUAPNG
|
7.3 | IC50 | 2 | — | |
DLUHYYWDKTVUNT
|
7.3 | IC50 | 2 | — | |
DPUCGDIRADRVPW
|
7.3 | IC50 | 2 | — | |
DXTPGWQAXLDDNL
|
7.3 | IC50 | 2 | — | |
FEAUSMUUPSCPKO
|
7.3 | IC50 | 2 | — | |
FGASSPDBSDOEPX
|
7.3 | IC50 | 2 | — | |
FGBWUXHBTBMVKE
|
7.3 | IC50 | 2 | — | |
FICRVLXLXMNVDH
|
7.3 | IC50 | 2 | — | |
FJBDTVHTQZMFJX
|
7.3 | IC50 | 2 | — | |
FMVABZINBVIDQL
|
7.3 | IC50 | 2 | — | |
FOIMBMUQCPZLMT
|
7.3 | IC50 | 2 | — | |
FOUDITGFIOIXRN
|
7.3 | IC50 | 2 | — | |
FROVAICQVUYMQU
|
7.3 | IC50 | 2 | — | |
FSVDYFNASNQHCE
|
7.3 | IC50 | 2 | — | |
FSVDYFNASNQHCE
|
7.3 | IC50 | 2 | — | |
FUOCXMOMJRLFAS
|
7.3 | IC50 | 2 | — | |
FUYXWABFTBBPPQ
|
7.3 | IC50 | 2 | — | |
FVNHWMOCBZQTBI
|
7.3 | IC50 | 2 | — | |
GANBXEQLAOHECS
|
7.3 | IC50 | 2 | — | |
GFARMNLPSPHGIR
|
7.3 | IC50 | 2 | — | |
GFQRQKUOFVNFKW
|
7.3 | IC50 | 2 | — | |
GIPUEKGFFDJJJJ
|
7.3 | IC50 | 2 | — | |
GJIAQUPOXRGEOW
|
7.3 | IC50 | 2 | — | |
GNGJWPZEJKPGFY
|
7.3 | IC50 | 2 | — | |
GNXFBTOJIPLCGB
|
7.3 | IC50 | 2 | — | |
GSJYABPCKQDTOX
|
7.3 | IC50 | 2 | — | |
GXKFLWFIKGXVFH
|
7.3 | IC50 | 2 | — | |
HBNAUONLWDFYEA
|
7.3 | IC50 | 2 | — | |
HKVJGRGOCHBUFK
|
7.3 | IC50 | 2 | — | |
HKVJGRGOCHBUFK
|
7.3 | IC50 | 2 | — | |
HKVJGRGOCHBUFK
|
7.3 | IC50 | 2 | — | |
HMFIFAOORJCVCB
|
7.3 | IC50 | 2 | — | |
HPTOTBDEYJWXMS
|
7.3 | IC50 | 2 | — | |
HQLFULDUYCCJPE
|
7.3 | IC50 | 2 | — | |
HRXPLCSOQNEFRZ
|
7.3 | IC50 | 2 | — | |
HSPMCXSTLBKXFP
|
7.3 | IC50 | 2 | — |