Target Details
UniProt ACQ14145
Gene SymbolKEAP1
Protein NameKelch-like ECH-associated protein 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF07707 (BACK) PF00651 (BTB) PF01344 (Kelch_1) PF24681 (Kelch_KLHDC2_KLHL20_DRC7)
Summary
  • Multi-target molecules 558
  • Clinical molecules 0
  • Avg pChEMBL 7.21
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (558)
InChIKey pChEMBL Type Targets Clinical
KFORSHXZAGQBCD 7.8 Kd 2
JJOFXZVJJGEQCK 7.8 IC50 2
FQVLNJYKCWMFHE 7.8 Kd 2
NEQJHAQENWACJE 7.8 Kd 2
QUJAHTSGLDPGHW 7.8 IC50 2
WQIYQSZCGZPQSX 7.8 IC50 2
YXZYLROMQQGNAT 7.8 Kd 2
NAUNGQVWVDFCQT 7.7 IC50 2
ZDUXQRUQCLUZNW 7.7 Kd 2
KFORSHXZAGQBCD 7.7 Kd 2
AHNXOLRIYAUDAJ 7.7 Kd 2
YXZYLROMQQGNAT 7.7 Kd 2
IMRNAESQPBZZKY 7.7 Kd 2
RWPONSQQBPIJRE 7.7 IC50 2
VWVMLPGRONCTQT 7.7 IC50 2
LFSYTNSCKJHRHR 7.6 IC50 2
RSKHAKDCRLZRNZ 7.6 Kd 2
KWSIQJUNYMMCTB 7.6 IC50 2
JTDWZQZKKFDOFM 7.6 Kd 2
WGYGFQFSIPMBHW 7.6 IC50 2
WVIVHXXSXLPJSU 7.6 IC50 2
BZBMUGXSZACOTM 7.5 Kd 2
FXADTNLKEANMJS 7.5 IC50 2
PWKJRVHFVZDUJL 7.5 Kd 2
REZAVPKMKABZLC 7.5 IC50 2
LUWNQRCIIOOCLS 7.5 IC50 2
ZDNGJXBUEQNFBQ 7.5 IC50 2
SNLIUNXULFSSAY 7.5 IC50 2
MZSWYXRPAMGWQY 7.4 IC50 2
BLJRYRIUUYNZFT 7.4 Ki 2
PMPKZTLVXIBPDN 7.4 Ki 2
RSPIKPFHLPIDKV 7.4 IC50 2
NTHLVVMPSHXUER 7.4 IC50 2
XEACSCDYNLDUDF 7.4 IC50 2
KDPCJWPUWRBBQU 7.3 IC50 2
IJHWQGAWCBWPSG 7.3 IC50 2
RTGHTXKISWZXKJ 7.3 IC50 2
GMVHZYNTLZSZQE 7.3 IC50 2
JAVOONPTJYTDCV 7.3 IC50 2
ZDNGJXBUEQNFBQ 7.3 IC50 2
PWKJRVHFVZDUJL 7.3 Kd 2
GAFLTUQDNVDCCP 7.3 Ki 2
LPKUZUTXBLBZSN 7.3 IC50 2
MTEYUVLCMWDLCD 7.3 IC50 2
NAIGTYLAELHHHM 7.3 Kd 2
SNWXNMFUFJGUTF 7.3 IC50 2
ZUIXHSIMKQZYPV 7.3 Kd 2
AKHCBMLHZMAGJM 7.3 IC50 2
BIHHECVWYUSKTL 7.3 IC50 2
BKKIQOWFHQPZEE 7.3 IC50 2
2D structure