Target Details
UniProt ACQ14145
Gene SymbolKEAP1
Protein NameKelch-like ECH-associated protein 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF07707 (BACK) PF00651 (BTB) PF01344 (Kelch_1) PF24681 (Kelch_KLHDC2_KLHL20_DRC7)
Summary
  • Multi-target molecules 558
  • Clinical molecules 0
  • Avg pChEMBL 7.21
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (558)
InChIKey pChEMBL Type Targets Clinical
LMQUBMLJZUWJRA 8.7 Kd 2
MCNYDHMNNGQZKU 8.7 Kd 2
SEYURAKXESNAMM 8.7 Kd 2
FCNFVOASVAFDIA 8.7 Kd 2
NVTPQMGCGHVFCU 8.7 Kd 2
FUSGWTIAPSLBBU 8.7 Kd 2
XUTKOLZVFVMAAY 8.7 Kd 2
IVSJVQZQYUVWHY 8.7 Kd 2
IWQYKEFJRDQJID 8.7 Kd 2
JEKSABWNOURZQX 8.6 Kd 2
KZCCKWDMRUQZRK 8.6 Kd 2
QXGZEGRFLMINNB 8.6 Kd 2
GZEVURFUHFYNDN 8.6 Kd 2
SOXOJUYWHVRMEF 8.6 Kd 2
DPBPSWZEKFMRIP 8.6 Kd 2
QTKISLYKZJKIKD 8.6 Kd 2
SPSYSXPCMXKWMY 8.6 Kd 2
CIQCGEVOKCUAIQ 8.6 Kd 2
MCDUEENZHCKFFC 8.6 Kd 2
XUTKOLZVFVMAAY 8.5 Kd 2
NXHZXXCSLXFYDJ 8.5 Kd 2
PRDCMJBDOVGICT 8.4 Kd 2
KMHWCKHBMPPAGF 8.4 Kd 2
QTKISLYKZJKIKD 8.4 Kd 2
VGAUNNBMILDZOW 8.4 Kd 2
RKHNUOKYCVBCRZ 8.3 Kd 2
HBYJPCOLBXNUQX 8.3 Kd 2
FCUHBMJCDSGVHP 8.3 Kd 2
YUTXJSZCUZEBPT 8.2 Kd 2
MCNYDHMNNGQZKU 8.2 Kd 2
OLLUZVHWYUYFAK 8.2 IC50 2
NKAJSIIDIPWQJJ 8.2 Kd 2
JNAMGNWTFMLHQC 8.2 IC50 2
TZTAISDLASISEW 8.2 IC50 2
IHLRKIWSZPXPKS 8.1 IC50 2
FCUHBMJCDSGVHP 8.1 Kd 2
DPBPSWZEKFMRIP 8.1 Kd 2
ASPKWDYARXRMAC 8.1 Kd 2
AYIQSLPGRXOWNY 8.1 Kd 2
ULCMDORLNFVULD 8.0 IC50 2
BVWKAUMFAYUKCN 8.0 IC50 2
GZEVURFUHFYNDN 8.0 Kd 2
VZVCHNYRESPRBX 8.0 IC50 2
PWTZMRSNENLEFH 7.9 IC50 2
HSKNRAQRJUMEIL 7.9 IC50 2
ITJMUCNXRCRSBV 7.9 Kd 2
PJEFMHSQDYYADJ 7.9 IC50 2
FYOHBNAOGGBOGT 7.9 IC50 2
CIQCGEVOKCUAIQ 7.9 Kd 2
NRGDPQSGSQBMPD 7.9 IC50 2
2D structure