Target Details
| UniProt AC | Q14145 |
|---|---|
| Gene Symbol | KEAP1 |
| Protein Name | Kelch-like ECH-associated protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07707 (BACK) PF00651 (BTB) PF01344 (Kelch_1) PF24681 (Kelch_KLHDC2_KLHL20_DRC7) |
Summary
- Multi-target molecules 558
- Clinical molecules 0
- Avg pChEMBL 7.21
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (558)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YXLKLSNRFCRSCM
|
6.0 | IC50 | 2 | — | |
ZAYWCPWPNQTOJO
|
6.0 | IC50 | 2 | — | |
AUTGDVUDNHXSHF
|
6.0 | IC50 | 2 | — | |
AYFVRYXNDHBECD
|
6.0 | Kd | 2 | — | |
CJHZLORMVFKACE
|
6.0 | IC50 | 2 | — | |
DXNNXGUWLIVFDR
|
6.0 | Kd | 2 | — | |
FRRZRAZHHYLGGZ
|
6.0 | IC50 | 2 | — | |
PKFCZHGGONJKQF
|
6.0 | IC50 | 2 | — |