Target Details
| UniProt AC | Q14145 |
|---|---|
| Gene Symbol | KEAP1 |
| Protein Name | Kelch-like ECH-associated protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07707 (BACK) PF00651 (BTB) PF01344 (Kelch_1) PF24681 (Kelch_KLHDC2_KLHL20_DRC7) |
Summary
- Multi-target molecules 558
- Clinical molecules 0
- Avg pChEMBL 7.21
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (558)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GYFMCCVPZGXQPI
|
6.2 | Ki | 2 | — | |
WLXLBNHWWYEQCG
|
6.2 | IC50 | 2 | — | |
XGGQQFHSICPQPI
|
6.2 | Kd | 2 | — | |
ADFGTGZXVNHSHG
|
6.2 | Kd | 2 | — | |
ASEIYZQTQCPTHI
|
6.2 | Ki | 2 | — | |
ZWLXITPIUVTPDI
|
6.2 | IC50 | 2 | — | |
LAXJJFZYISZHTH
|
6.2 | Kd | 2 | — | |
PHZBSENPMPRYCX
|
6.2 | IC50 | 2 | — | |
WOTGMDIMMYQXRU
|
6.2 | IC50 | 2 | — | |
XTQMICBWPLVONW
|
6.2 | IC50 | 2 | — | |
SDCHEHCCVZBOPQ
|
6.2 | Ki | 2 | — | |
TYRJUXNRNRLVEE
|
6.2 | IC50 | 2 | — | |
YVLLANYGJMGXEE
|
6.2 | Kd | 2 | — | |
ZFAWWQNTBJRYJU
|
6.2 | Ki | 2 | — | |
GXSFTGVLOAKALY
|
6.2 | IC50 | 2 | — | |
XLUSKTXXBQNSSG
|
6.2 | IC50 | 2 | — | |
IUQICDGBODPWAB
|
6.2 | Ki | 2 | — | |
XUKXFTLJLIEKKZ
|
6.2 | Kd | 2 | — | |
ZWVUKRKRSHBJQP
|
6.2 | Kd | 2 | — | |
ZPWOSQULANINNR
|
6.2 | IC50 | 2 | — | |
RLXZLIPXEZYRSP
|
6.2 | Kd | 2 | — | |
JWDSRPNRRATQKY
|
6.1 | Kd | 2 | — | |
SAPJYRTVXRKYMQ
|
6.1 | Ki | 2 | — | |
AWFONHWHPMHOEM
|
6.1 | IC50 | 2 | — | |
IDDVVOGRPYQGJG
|
6.1 | IC50 | 2 | — | |
PPAVPTUSMNPROA
|
6.1 | IC50 | 2 | — | |
YTUXAQFRBNUADX
|
6.1 | IC50 | 2 | — | |
YTUXAQFRBNUADX
|
6.1 | IC50 | 2 | — | |
DLKNSOBRFKAQHY
|
6.1 | Ki | 2 | — | |
LNENLABLFGGAFF
|
6.1 | IC50 | 2 | — | |
OXPMJRFVNJYLMF
|
6.1 | IC50 | 2 | — | |
VRFYWLIHNVOIDV
|
6.1 | IC50 | 2 | — | |
XZIIWNBFZABURQ
|
6.1 | Kd | 2 | — | |
YWENUUZTMLXNIY
|
6.1 | IC50 | 2 | — | |
SZAQVULLZNMZEI
|
6.1 | Kd | 2 | — | |
AAHBRGHGLGSULN
|
6.1 | Kd | 2 | — | |
DPCJVXCKIOCDNF
|
6.1 | IC50 | 2 | — | |
KMLNCQNKHLOHEL
|
6.1 | IC50 | 2 | — | |
SFFSAQRGKZSDJN
|
6.1 | IC50 | 2 | — | |
ZELWYLZRAFSOOR
|
6.1 | Kd | 2 | — | |
YHBYNIAFTHBNFW
|
6.1 | IC50 | 2 | — | |
FDKHUGAIEHHSKD
|
6.0 | IC50 | 2 | — | |
XHXHGTBWDVNVCU
|
6.0 | IC50 | 2 | — | |
GLCJZDMESDJEPO
|
6.0 | IC50 | 2 | — | |
YGORVLIVECUGIV
|
6.0 | IC50 | 2 | — | |
BIPORTLLFPOICC
|
6.0 | IC50 | 2 | — | |
IAUPZZWJUFVQJA
|
6.0 | IC50 | 2 | — | |
MBXJNJNZSJKACU
|
6.0 | IC50 | 2 | — | |
NHYBXSMAVMJFIN
|
6.0 | IC50 | 2 | — | |
SSGZMSYLGMICAH
|
6.0 | IC50 | 2 | — |