Target Details
| UniProt AC | Q14145 |
|---|---|
| Gene Symbol | KEAP1 |
| Protein Name | Kelch-like ECH-associated protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07707 (BACK) PF00651 (BTB) PF01344 (Kelch_1) PF24681 (Kelch_KLHDC2_KLHL20_DRC7) |
Summary
- Multi-target molecules 558
- Clinical molecules 0
- Avg pChEMBL 7.21
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (558)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BTPDPSLUOKOLFC
|
6.3 | IC50 | 2 | — | |
CAJHFKZCUUGUSQ
|
6.3 | IC50 | 2 | — | |
CCKFFZWASQCQFD
|
6.3 | IC50 | 2 | — | |
CPQNNJBTSHDTLZ
|
6.3 | IC50 | 2 | — | |
CUENPUOZILZXSI
|
6.3 | IC50 | 2 | — | |
CXZPRQFTYURHET
|
6.3 | IC50 | 2 | — | |
DRSUZWSVWLQHEW
|
6.3 | IC50 | 2 | — | |
FGIULSJBSODLAD
|
6.3 | IC50 | 2 | — | |
FKGLABWENBSNRH
|
6.3 | IC50 | 2 | — | |
FRBDZDVSXHHBHW
|
6.3 | IC50 | 2 | — | |
FRPGONVMQZYDCC
|
6.3 | IC50 | 2 | — | |
GFARMNLPSPHGIR
|
6.3 | IC50 | 2 | — | |
GFARMNLPSPHGIR
|
6.3 | IC50 | 2 | — | |
GSFAKWDVAVVJHY
|
6.3 | IC50 | 2 | — | |
HTZLVFKYHDOFIL
|
6.3 | IC50 | 2 | — | |
JBQFMPMORHDMHZ
|
6.3 | IC50 | 2 | — | |
JWCCGAXRMNTCEB
|
6.3 | IC50 | 2 | — | |
JXCOERQLGLXVIK
|
6.3 | IC50 | 2 | — | |
KXTXQGKARMHJOC
|
6.3 | IC50 | 2 | — | |
LALJNFCDDXCGMH
|
6.3 | IC50 | 2 | — | |
LLMYBSXAZDMMIK
|
6.3 | IC50 | 2 | — | |
MDMOGTPMLUHGBG
|
6.3 | IC50 | 2 | — | |
MQSQNZXYSKOZIF
|
6.3 | IC50 | 2 | — | |
NICLDNFOUWEYPY
|
6.3 | IC50 | 2 | — | |
NICLDNFOUWEYPY
|
6.3 | IC50 | 2 | — | |
OYZIJXYHWRIKIW
|
6.3 | IC50 | 2 | — | |
PCWFDFLFSSELHV
|
6.3 | IC50 | 2 | — | |
PFCGOQHTVTVEGR
|
6.3 | IC50 | 2 | — | |
PRDDRPQTESJCMJ
|
6.3 | IC50 | 2 | — | |
PRPJMTIHQARBAD
|
6.3 | IC50 | 2 | — | |
QHHJBFGEOQGEIC
|
6.3 | IC50 | 2 | — | |
QLBKVJGMFUFAFO
|
6.3 | IC50 | 2 | — | |
RRSZSRNHVNNEPA
|
6.3 | IC50 | 2 | — | |
SINSEALUHHRXQF
|
6.3 | IC50 | 2 | — | |
SRMMWYRXUWFSNL
|
6.3 | IC50 | 2 | — | |
TYEFYUBZAKPDAX
|
6.3 | IC50 | 2 | — | |
UANMOFVJIKFJJT
|
6.3 | IC50 | 2 | — | |
UGALCWYPMZIMJQ
|
6.3 | IC50 | 2 | — | |
UOLHWQPOVKEGJH
|
6.3 | IC50 | 2 | — | |
UVNADZWWOXEWFH
|
6.3 | IC50 | 2 | — | |
VLUCKJQHVVDJRS
|
6.3 | IC50 | 2 | — | |
WMFNTTPHZCWVFH
|
6.3 | IC50 | 2 | — | |
XDOGAMNAMXXKOO
|
6.3 | IC50 | 2 | — | |
XGHQHSHDBJZAOQ
|
6.3 | IC50 | 2 | — | |
XKXXEUFAYDHYPN
|
6.3 | IC50 | 2 | — | |
YFUKZAAYGLSBNI
|
6.3 | IC50 | 2 | — | |
ZHMFLGKJTRLMKZ
|
6.3 | IC50 | 2 | — | |
IEYJKFLEKQWEPR
|
6.2 | Kd | 2 | — | |
MFYPHSBKCCZZFC
|
6.2 | IC50 | 2 | — | |
CYYUUKBJPMWCSI
|
6.2 | IC50 | 2 | — |