Target Details
| UniProt AC | Q14012 |
|---|---|
| Gene Symbol | CAMK1 |
| Protein Name | Calcium/calmodulin-dependent protein kinase type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 26
- Clinical molecules 2
- Avg pChEMBL 6.79
KEGG Pathways (4)
Active Molecules (26)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RJTDRNOTQRMDCY
|
8.7 | IC50 | 4 | — | |
BWBUPDTUXQDHSX
|
8.5 | IC50 | 5 | — | |
HKSZLNNOFSGOKW
|
7.9 | Ki | 118 | — | |
HKSZLNNOFSGOKW
|
7.6 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
7.6 | Kd | 213 | — | |
GHPFQRTVUDXWCC
|
7.5 | Ki | 35 | — | |
CFIBXVQLBVNOHW
|
7.1 | Ki | 64 | — | |
NJPWCTYVEJIQBM
|
7.0 | Ki | 72 | — | |
BPNUQXPIQBZCMR
|
6.9 | Ki | 60 | — | |
UIARLYUEJFELEN
|
6.9 | Kd | 289 | Yes | |
XJSFDMGICAWQFS
|
6.7 | Ki | 60 | — | |
NHHQJBCNYHBUSI
|
6.6 | Kd | 220 | — | |
CHTMRWQLNNRRFJ
|
6.6 | Ki | 70 | — | |
MVJMMLFMPWITEJ
|
6.5 | Ki | 110 | — | |
OWRXHGAFWZFFCW
|
6.5 | Ki | 113 | — | |
VXYDJXMHISGSDA
|
6.5 | Ki | 59 | — | |
NFKMFNBKEOQNPZ
|
6.4 | Ki | 43 | — | |
HFNKQEVNSGCOJV
|
6.3 | Kd | 65 | — | |
UMTWTCVTRDYHQQ
|
6.3 | Ki | 56 | — | |
JZTOUVBEZONDKA
|
6.2 | Ki | 80 | — | |
FLEAYYMORDPWAJ
|
6.1 | Ki | 90 | — | |
NRZYTPAJGVTKIM
|
6.1 | Ki | 38 | — | |
WINHZLLDWRZWRT
|
6.0 | Kd | 201 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JZSWBZHJDCDLHK
|
6.0 | Ki | 10 | — | |
WPHKIQPVPYJNAX
|
6.0 | Ki | 81 | — |