Target Details
| UniProt AC | Q13976 |
|---|---|
| Gene Symbol | PRKG1 |
| Protein Name | cGMP-dependent protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF16808 (PKcGMP_CC) PF00069 (Pkinase) |
Summary
- Multi-target molecules 135
- Clinical molecules 11
- Avg pChEMBL 6.99
KEGG Pathways (11)
Associated Diseases (1)
Active Molecules (135)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZWVZORIKUNOTCS
|
6.4 | Ki | 69 | — | |
QQWUGDVOUVUTOY
|
6.4 | Kd | 231 | Yes | |
ZKZXNDJNWUTGDK
|
6.3 | Ki | 9 | — | |
DBKQWGCVGCVPIP
|
6.3 | Ki | 21 | — | |
MASJMHFQMYAPJR
|
6.3 | Ki | 41 | — | |
MIYRKQLKDQNUKZ
|
6.3 | Ki | 23 | — | |
QAJPIJHWTGPUNZ
|
6.3 | Ki | 37 | — | |
QPORZABOFXPRHM
|
6.3 | Ki | 18 | — | |
YKJSWMAVAKRUAN
|
6.3 | Ki | 19 | — | |
YKYRQCWLYUTVIE
|
6.3 | Ki | 16 | — | |
WVGDUQVQWLHVEA
|
6.2 | IC50 | 4 | — | |
BEJGILHFZNTYCX
|
6.2 | Ki | 7 | — | |
DWTNLZZEPSCAIH
|
6.2 | Ki | 25 | — | |
ISEDKXOMRIKZPK
|
6.2 | Ki | 13 | — | |
VIJBEUTVNBPGIU
|
6.2 | Ki | 19 | — | |
WYLVFMBGPRCDQF
|
6.2 | Ki | 14 | — | |
XJVDVWLKPCDPAA
|
6.2 | Kd | 3 | — | |
YVKVSKQNYIHXPX
|
6.2 | Ki | 7 | — | |
ZGZVRPRSFXRGCF
|
6.2 | Ki | 76 | — | |
DHYYPPHQZMSVKX
|
6.1 | Ki | 2 | — | |
CLEGDJQQHUTCOW
|
6.1 | Ki | 43 | — | |
FDBPGAHVEGEARY
|
6.1 | Ki | 19 | — | |
JJJSCYSPSKBQAX
|
6.1 | Ki | 34 | — | |
KAKGFGCTONHQJW
|
6.1 | Ki | 25 | — | |
OAVGBZOFDPFGPJ
|
6.1 | Ki | 42 | Yes | |
RKUKAACYUCUJEE
|
6.1 | Ki | 58 | — | |
SPMHGQZFMNZCBV
|
6.1 | Ki | 30 | Yes | |
XAHJIRNRDAKTEF
|
6.1 | Ki | 18 | — | |
ZLVOTRRGLSDLPF
|
6.1 | Ki | 36 | — | |
AWDORCFLUJZUQS
|
6.0 | Ki | 22 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JCFJQIHDZHHMQT
|
6.0 | Ki | 42 | — | |
PAIFYAZSILXLBO
|
6.0 | Ki | 26 | — | |
UTQPKPHUIMHAAN
|
6.0 | Ki | 22 | — | |
YPJJSXBVVGPFHA
|
6.0 | Ki | 18 | — |