Target Details
UniProt ACQ13976
Gene SymbolPRKG1
Protein NamecGMP-dependent protein kinase 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00027 (cNMP_binding) PF16808 (PKcGMP_CC) PF00069 (Pkinase)
Summary
  • Multi-target molecules 135
  • Clinical molecules 11
  • Avg pChEMBL 6.99
Top Co-occurrence Targets
Active Molecules (135)
InChIKey pChEMBL Type Targets Clinical
ADMFLILDQJSEIK 7.0 Ki 72
FUMCKNCUEAQHCV 7.0 Ki 103
OEEGUWWPGAZRIJ 7.0 Ki 21
SYSUZXPGQXEWCZ 7.0 Ki 10
ZKHDDJKHTPLPOQ 7.0 Ki 62
ZRQXCQXWTLVASO 7.0 Ki 36
NXSJMRCTGYTSTK 7.0 Kd 200
ASNQMAVHHGGQRB 6.9 Ki 14
FQEODTMNWMDUMD 6.9 Ki 25
GCYXEGSPUDSZJY 6.9 Ki 82
HXDDWVMJYDULAZ 6.9 Ki 13
NEWAULHLLUCDPD 6.9 Ki 27
KGPGFQWBCSZGEL 6.9 Kd 59 Yes
BPNUQXPIQBZCMR 6.8 Ki 60
KWRXWPRFIUJQBP 6.8 Ki 25
SBFPHSVZEXSHTL 6.8 Ki 62
VVQQRUZZQQSDEI 6.8 Ki 6
XPHWIERLJBFPFV 6.8 Ki 69
YOVNFNXUCOWYSG 6.8 Ki 33 Yes
CLRFYTGANQZOBS 6.7 Ki 41
DPPIQOOVRLCHQC 6.7 Ki 6
MBRVCJRFWYHVHE 6.7 Ki 9
TVEREFRWBLRPPJ 6.7 Ki 15
VUHZDNOPEVGHEO 6.7 Ki 29
XFWUTMHVDGPWLH 6.7 Ki 75
BMGQWWVMWDBQGC 6.6 Kd 147 Yes
MIKAKZKNMYZLDX 6.6 Ki 42
RFVBRKXQYUDGIO 6.6 Ki 23
SOVYWBOZOBVFLP 6.6 Ki 10
TWCARTFPHQNBPF 6.6 Ki 16
UTFXYGYVDDLJER 6.6 Ki 36
YWTBGJGMTBHQTM 6.6 Ki 65
ZMBDLCDLIZXFHY 6.6 Ki 9
ZYTFPHRVOZXPGZ 6.6 Ki 30
BPNUQXPIQBZCMR 6.6 Kd 83 Yes
JDUBGYFRJFOXQC 6.5 Kd 13
CZIGMBNEFWBEMD 6.5 Ki 16
HZBPSQIDFQPUKG 6.5 IC50 2
JSKUWFIZUALZLX 6.5 Ki 33
KCKXYZOBGBJZEG 6.5 Ki 36
KXPWWMPXNUOYOH 6.5 Ki 24
ORUUEFDGYYTXAF 6.5 Ki 26
UDFDIIVNIYWXDM 6.5 Ki 74
XBDWKVLCDCUNHH 6.5 Ki 18
XSDJOIOVIMPMHD 6.5 Ki 44
XSRHBCYNCKAFKS 6.5 Ki 45
UIARLYUEJFELEN 6.4 Kd 289 Yes
IJNGXROUMFEKDB 6.4 Ki 39
LWBSSNRDDDFHSH 6.4 Ki 9
MADCXGNPDBWPLM 6.4 Ki 25
2D structure