Target Details
| UniProt AC | Q13946 |
|---|---|
| Gene Symbol | PDE7A |
| Protein Name | High affinity 3',5'-cyclic-AMP phosphodiesterase 7A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00233 (PDEase_I) |
Summary
- Multi-target molecules 157
- Clinical molecules 0
- Avg pChEMBL 7.59
KEGG Pathways (3)
Active Molecules (157)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LMANVTDDCGUCNF
|
7.3 | IC50 | 2 | — | |
JMCCOEJBVQAXPU
|
7.3 | IC50 | 2 | — | |
GURINCBMWKPPBD
|
7.3 | IC50 | 2 | — | |
ILHCAAUBKXDWAM
|
7.2 | IC50 | 2 | — | |
AITIZXXDRMMFPO
|
7.2 | IC50 | 2 | — | |
FWQKUKGUXLHLLO
|
7.2 | IC50 | 2 | — | |
HNDKBWFZQQACDL
|
7.2 | IC50 | 2 | — | |
LQTUFULCEXRYTR
|
7.2 | IC50 | 2 | — | |
OGCNKFMAMJTOMD
|
7.2 | IC50 | 2 | — | |
QSLZYOAQCXNUMC
|
7.2 | IC50 | 2 | — | |
SLFAGMLIYQWDMX
|
7.2 | IC50 | 2 | — | |
ULGCVTFBIMJXBI
|
7.2 | IC50 | 2 | — | |
XLPVHHYXTYQBMA
|
7.2 | IC50 | 2 | — | |
YGYWQAJIPHCBLS
|
7.2 | IC50 | 2 | — | |
YXBFNVYLMDJRLF
|
7.2 | IC50 | 2 | — | |
YPZRKHZFHQJVDJ
|
7.2 | IC50 | 2 | — | |
WNKDNKJGTZVRBX
|
7.1 | IC50 | 2 | — | |
XAIXRJONTNTVTN
|
7.1 | IC50 | 2 | — | |
JELWUFXWZSYANR
|
7.1 | IC50 | 2 | — | |
IFIUFCJFLGCQPH
|
7.0 | IC50 | 2 | — | |
HMLIQWYFUWNFED
|
7.0 | IC50 | 2 | — | |
GMUIDKJUSNEWSL
|
7.0 | IC50 | 2 | — | |
VTPBHYIYWZNATF
|
6.9 | IC50 | 2 | — | |
PPFGVIYVXGCXRU
|
6.8 | IC50 | 3 | — | |
RTVAXMAAIDVFHH
|
6.8 | IC50 | 2 | — | |
JYCHFFXFIDUIDW
|
6.8 | IC50 | 2 | — | |
WQQNYFFWISBZNB
|
6.7 | IC50 | 2 | — | |
VIQYGEOSRSOQKW
|
6.6 | Ki | 3 | — | |
FNTGJJLOKISHIS
|
6.6 | IC50 | 3 | — | |
PMOGXWRUBZRFGT
|
6.6 | Ki | 3 | — | |
IWQJRWQPBCCRGZ
|
6.5 | IC50 | 8 | — | |
OVSHRJGAYOZGQR
|
6.5 | IC50 | 8 | — | |
OGVUDOFPSURVMY
|
6.5 | IC50 | 2 | — | |
RGPAMUDSBRASGW
|
6.5 | IC50 | 2 | — | |
OFZGCAMFVYIIHV
|
6.5 | IC50 | 24 | — | |
RMKFHXBPLKSLMZ
|
6.5 | IC50 | 3 | — | |
AXNJNPPDLFAOFG
|
6.3 | Ki | 2 | — | |
BFNBJSXMXXQLAW
|
6.3 | IC50 | 2 | — | |
NUMTXTPCPDSVTH
|
6.3 | IC50 | 2 | — | |
MVPONTPZYKDJPY
|
6.3 | IC50 | 3 | — | |
RAQWULABCGLUNW
|
6.3 | IC50 | 2 | — | |
BTYONSNIAIDRLB
|
6.3 | Ki | 3 | — | |
DJJOAJCVIYRELX
|
6.3 | IC50 | 2 | — | |
IZEKFCXSFNUWAM
|
6.2 | Ki | 19 | — | |
CYERGDRLLOCHQC
|
6.2 | Ki | 3 | — | |
JEWCYYAOLPVLHO
|
6.2 | IC50 | 3 | — | |
QHLZYKWHQKCZMD
|
6.2 | IC50 | 3 | — | |
QHNOASMPSYWQOJ
|
6.2 | IC50 | 2 | — | |
KOVUQUXRMIAWMX
|
6.2 | IC50 | 3 | — | |
USZAGAREISWJDP
|
6.1 | IC50 | 7 | — |