Target Details
| UniProt AC | Q13946 |
|---|---|
| Gene Symbol | PDE7A |
| Protein Name | High affinity 3',5'-cyclic-AMP phosphodiesterase 7A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00233 (PDEase_I) |
Summary
- Multi-target molecules 157
- Clinical molecules 0
- Avg pChEMBL 7.59
KEGG Pathways (3)
Active Molecules (157)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UJLHNYPXKZJKLV
|
10.0 | IC50 | 24 | — | |
KXCOKRBRUWINCT
|
9.9 | IC50 | 24 | — | |
KPFFPWNKWSYQFT
|
9.8 | IC50 | 24 | — | |
GOBQSCBEINUNFL
|
9.6 | IC50 | 24 | — | |
AFCWMWBOATWMJV
|
9.5 | IC50 | 24 | — | |
DKSKKVAOIPURFT
|
9.5 | IC50 | 24 | — | |
OZGMVFAOJFAKML
|
9.5 | IC50 | 3 | — | |
XSNLHLHGJSLJQA
|
9.2 | IC50 | 4 | — | |
AWDJJMXJUOHGLC
|
9.1 | IC50 | 3 | — | |
BPBDCOLBZYWXHD
|
9.0 | IC50 | 24 | — | |
FMMIDZWTNQYEIY
|
9.0 | IC50 | 24 | — | |
JUTYAJADZTZCBP
|
9.0 | IC50 | 2 | — | |
HQKUXNBKAFHBHJ
|
9.0 | IC50 | 2 | — | |
DVOSPTOWEQEYQB
|
8.9 | IC50 | 3 | — | |
MEQLCCSBIKIYJU
|
8.9 | IC50 | 2 | — | |
JUDJZYCORAYMNM
|
8.8 | IC50 | 2 | — | |
LDDQCPUHJNDZLS
|
8.8 | IC50 | 2 | — | |
ZRXCXSQNKXCJNQ
|
8.8 | IC50 | 2 | — | |
WYFACFDIJBGSEA
|
8.7 | IC50 | 2 | — | |
XOHAWIWJMGSBAH
|
8.7 | IC50 | 2 | — | |
XFJQWGBAKVNZJJ
|
8.6 | IC50 | 2 | — | |
FIUCLBJMUGCQTF
|
8.6 | IC50 | 8 | — | |
NLFMMOQCAASWGC
|
8.6 | IC50 | 2 | — | |
OSIAQFSEAYCSKV
|
8.5 | IC50 | 6 | — | |
FTTARRILKZGDNU
|
8.5 | IC50 | 5 | — | |
AABLQBRGBFMNIT
|
8.4 | IC50 | 2 | — | |
ORDCDFJDRJJITQ
|
8.4 | IC50 | 5 | — | |
UZUDVFPSKOVACF
|
8.4 | IC50 | 2 | — | |
TZXUAKHZPAHOMA
|
8.4 | IC50 | 2 | — | |
KRKCXJIRRPKWPM
|
8.3 | IC50 | 2 | — | |
KNKPONLBTNMNAZ
|
8.3 | IC50 | 2 | — | |
MEHFKIXPEUTUIO
|
8.3 | IC50 | 2 | — | |
VNAHXSARBLNPNV
|
8.3 | IC50 | 2 | — | |
QKFLLRFETHNLQD
|
8.3 | IC50 | 2 | — | |
AIOOOOYCTWPHCO
|
8.2 | IC50 | 2 | — | |
BBEQXRUPYAKWEQ
|
8.2 | IC50 | 2 | — | |
OIRJTQAINLCWJS
|
8.2 | IC50 | 2 | — | |
YGEGQTNEVVJOLB
|
8.2 | IC50 | 2 | — | |
RSTAFNGCTLDAPB
|
8.2 | IC50 | 2 | — | |
NAAQIZQJJJGURC
|
8.1 | IC50 | 2 | — | |
MZDYWLVQWRQFMV
|
8.0 | IC50 | 4 | — | |
OFWGHMAISKOSQV
|
8.0 | IC50 | 2 | — | |
UMKXDGBAQDPHBC
|
8.0 | IC50 | 2 | — | |
UNFGOVWIPVJXET
|
8.0 | IC50 | 2 | — | |
ZOSTZZLCBBHOHV
|
8.0 | IC50 | 5 | — | |
IGDJSSAOITZOHR
|
7.9 | IC50 | 2 | — | |
WUCGXMCXJRLPEJ
|
7.9 | IC50 | 2 | — | |
WZHFBTOHDLSCOL
|
7.9 | IC50 | 2 | — | |
DNHMCBAUCKMZOU
|
7.8 | IC50 | 2 | — | |
ZMZGFAGXALOLIK
|
7.8 | IC50 | 4 | — |