Target Details
| UniProt AC | Q13882 |
|---|---|
| Gene Symbol | PTK6 |
| Protein Name | Protein-tyrosine kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 146
- Clinical molecules 13
- Avg pChEMBL 7.1
Active Molecules (146)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ULTCRVJUAZCGPP
|
6.5 | IC50 | 5 | — | |
HXHAJRMTJXHJJZ
|
6.5 | Ki | 52 | Yes | |
TVLFEDKEAOXRCZ
|
6.5 | Ki | 22 | — | |
UOOZSMNSBYVUGZ
|
6.5 | Ki | 32 | — | |
VKBFHTIUXUCYRQ
|
6.5 | Ki | 66 | — | |
WMMNTQFZCHUZSM
|
6.5 | IC50 | 14 | — | |
RKBYYWVZFBATHQ
|
6.5 | IC50 | 12 | — | |
VTJHGMZHVOXJPG
|
6.5 | IC50 | 15 | — | |
MOSKATHMXWSZTQ
|
6.5 | IC50 | 16 | Yes | |
NHHQJBCNYHBUSI
|
6.4 | Kd | 220 | — | |
LYADGAGFYYXXIO
|
6.4 | IC50 | 82 | — | |
XKFTZKGMDDZMJI
|
6.4 | Ki | 56 | — | |
YEKVTSRZMPLPFK
|
6.4 | Ki | 17 | — | |
SIXVRXARNAVBTC
|
6.4 | IC50 | 12 | — | |
CNTCGRJDUJEUDG
|
6.3 | Ki | 37 | — | |
WFTZMAAMCVPJJT
|
6.3 | Ki | 26 | — | |
ZGDSBEUMPIMXBM
|
6.3 | Ki | 42 | — | |
ZKHDDJKHTPLPOQ
|
6.3 | Ki | 62 | — | |
DPZGKYJHTOSMIA
|
6.3 | IC50 | 8 | — | |
KZRDVFBPXXGSPD
|
6.3 | IC50 | 9 | — | |
QUFURWJAQILIFO
|
6.3 | IC50 | 9 | — | |
QYZOGCMHVIGURT
|
6.3 | Kd | 26 | Yes | |
OUKYUETWWIPKQR
|
6.2 | Kd | 31 | Yes | |
XXJWYDDUDKYVKI
|
6.2 | Kd | 52 | — | |
GQGMUKOYILWOIQ
|
6.2 | Ki | 25 | — | |
HEKAIDKUDLCBRU
|
6.2 | Ki | 20 | — | |
RYYNGWLOYLRZLK
|
6.2 | Ki | 104 | — | |
WKCFYOHIHUZMEB
|
6.2 | IC50 | 5 | — | |
XFWUTMHVDGPWLH
|
6.2 | Ki | 75 | — | |
CQFVDHNTTRWVQD
|
6.1 | Ki | 9 | — | |
FMPKTXNCNJCHCC
|
6.1 | Ki | 25 | — | |
KAKFXRYHYUPXSU
|
6.1 | Ki | 16 | — | |
LYNBNVBMAGDJRW
|
6.1 | Ki | 81 | — | |
SPMVMDHWKHCIDT
|
6.1 | Kd | 30 | — | |
XCHWBXBDZRJVDP
|
6.1 | Ki | 51 | — | |
LCVIRAZGMYMNNT
|
6.1 | Kd | 20 | — | |
MHPRNHAIPCKPIR
|
6.0 | IC50 | 5 | — | |
YVXSYYKMNOMLIT
|
6.0 | IC50 | 5 | — | |
XGALLCVXEZPNRQ
|
6.0 | IC50 | 39 | Yes | |
YRCHYHRCBXNYNU
|
6.0 | Kd | 13 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MFAQYJIYDMLAIM
|
6.0 | Kd | 130 | Yes | |
PTVPBWWDGZSEAF
|
6.0 | Ki | 63 | — | |
RAHBGWKEPAQNFF
|
6.0 | Kd | 26 | — |