Target Details
| UniProt AC | Q13882 |
|---|---|
| Gene Symbol | PTK6 |
| Protein Name | Protein-tyrosine kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 146
- Clinical molecules 13
- Avg pChEMBL 7.1
Active Molecules (146)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LSJWYMSFUWBGPN
|
7.3 | IC50 | 17 | — | |
VAARYSWULJUGST
|
7.3 | Kd | 119 | Yes | |
CDISOBGWDHAHGF
|
7.3 | IC50 | 16 | — | |
JNAHXDJEKAMVMC
|
7.3 | IC50 | 3 | — | |
UYJNQQDJUOUFQJ
|
7.3 | Ki | 68 | — | |
UORAPQCBWYIISR
|
7.3 | IC50 | 15 | — | |
UORAPQCBWYIISR
|
7.3 | IC50 | 13 | — | |
UORAPQCBWYIISR
|
7.3 | IC50 | 12 | — | |
UORAPQCBWYIISR
|
7.3 | IC50 | 6 | — | |
UQRCJCNVNUFYDX
|
7.3 | Kd | 27 | — | |
BAIXSQGNLALLTR
|
7.3 | IC50 | 4 | — | |
GMPQGWXPDRNCBL
|
7.3 | IC50 | 4 | — | |
IBCGPVVKHZXWNX
|
7.3 | IC50 | 7 | — | |
NJKRMPNUGZAMJN
|
7.3 | IC50 | 5 | — | |
NTVNACFXAFFJQX
|
7.3 | IC50 | 2 | — | |
QQHSTSLAVGUPKP
|
7.3 | IC50 | 3 | — | |
RAJLVDVCHMUAEY
|
7.3 | IC50 | 2 | — | |
VWDNDBICKRVFCP
|
7.3 | IC50 | 4 | — | |
XJGZXZXWDRLHBF
|
7.3 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
7.2 | IC50 | 92 | — | |
JUSWPUDQOKINJO
|
7.2 | IC50 | 16 | — | |
OPHSZSZDICRBPP
|
7.2 | IC50 | 16 | — | |
DAIZZWZDMLDKTD
|
7.2 | IC50 | 2 | — | |
MGGBYMDAPCCKCT
|
7.2 | Kd | 23 | — | |
MOHYPRXHKRXDSE
|
7.2 | IC50 | 8 | — | |
XYFZVVYVIFJBIS
|
7.2 | IC50 | 17 | — | |
AHBFBRPGNOVEBK
|
7.2 | IC50 | 11 | — | |
DONQOOXVVSQFSF
|
7.2 | IC50 | 2 | — | |
SHPFDGWALWEPGS
|
7.2 | Kd | 35 | — | |
LAJAFFLJAJMYLK
|
7.1 | IC50 | 17 | — | |
LAUHLGUSVSJYCI
|
7.1 | IC50 | 16 | — | |
OWRXHGAFWZFFCW
|
7.1 | Ki | 113 | — | |
UUWNXFJBBYAMDT
|
7.1 | Ki | 46 | — | |
YZDJQTHVDDOVHR
|
7.1 | IC50 | 23 | — | |
OMIQRSKHABIPRH
|
7.1 | IC50 | 15 | — | |
BZBBQXMBSCKMNN
|
7.0 | IC50 | 2 | — | |
APPXQUDJLJXULP
|
7.0 | IC50 | 47 | — | |
GZYUJXFTHLKPAK
|
7.0 | IC50 | 16 | — | |
YHVHYWYQEFELOW
|
6.9 | IC50 | 44 | — | |
JSDGKSMNPHJDFK
|
6.9 | Ki | 35 | — | |
UHTHHESEBZOYNR
|
6.8 | Kd | 66 | Yes | |
HVXKQKFEHMGHSL
|
6.8 | Kd | 21 | — | |
WDTHDWKPTWWHLS
|
6.8 | IC50 | 13 | — | |
WOSKHXYHFSIKNG
|
6.8 | Kd | 24 | — | |
WKDACQVEJIVHMZ
|
6.8 | Kd | 46 | — | |
LOLPPWBBNUVNQZ
|
6.7 | Kd | 97 | Yes | |
HAYYBYPASCDWEQ
|
6.7 | IC50 | 47 | — | |
MVJMMLFMPWITEJ
|
6.7 | Ki | 110 | — | |
OSAWFUCUZJNEID
|
6.7 | IC50 | 20 | — | |
HKSZLNNOFSGOKW
|
6.6 | IC50 | 408 | — |