Target Details
| UniProt AC | Q13882 |
|---|---|
| Gene Symbol | PTK6 |
| Protein Name | Protein-tyrosine kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 146
- Clinical molecules 13
- Avg pChEMBL 7.1
Active Molecules (146)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CIGMIXWAESLRNR
|
8.7 | Kd | 5 | — | |
SFCBIFOAGRZJNX
|
8.7 | Kd | 22 | — | |
JSFCZQSJQXFJDS
|
8.6 | IC50 | 4 | — | |
FDVSOQRNTAPCHB
|
8.5 | Ki | 40 | — | |
MEQKJTZVPMNRIL
|
8.5 | IC50 | 2 | — | |
RXPZOSHFGJWSLQ
|
8.5 | IC50 | 6 | — | |
LCYSSHSIKSARGO
|
8.5 | IC50 | 19 | — | |
SSDFTYWIYVWCIE
|
8.5 | IC50 | 17 | — | |
AILRADAXUVEEIR
|
8.4 | IC50 | 75 | — | |
SEJGTFPOEJWEGG
|
8.4 | Kd | 149 | — | |
CEZMWLPQGCFDGW
|
8.3 | IC50 | 2 | — | |
GRLLIPLZODJAQA
|
8.3 | IC50 | 2 | — | |
XYFPWWZEPKGCCK
|
8.1 | IC50 | 34 | — | |
ZBNZXTGUTAYRHI
|
8.1 | IC50 | 102 | Yes | |
MIMOHMCANSGXIG
|
8.1 | IC50 | 15 | — | |
ZVPDNRVYHLRXLX
|
8.1 | Ki | 35 | Yes | |
PUKNKXZDTFQUDJ
|
8.0 | IC50 | 2 | — | |
HCVSOJQZDUYODJ
|
8.0 | IC50 | 2 | — | |
LVLFSSZNAIKYCD
|
8.0 | IC50 | 19 | — | |
FVHDMSVWNIOSFF
|
7.9 | IC50 | 2 | — | |
QODQEZHGGGAGFQ
|
7.9 | IC50 | 2 | — | |
GXJSLIOOPZRPEV
|
7.9 | Ki | 34 | — | |
MDTVHFCFGLWPLA
|
7.9 | IC50 | 2 | — | |
ZCIUSITUWMIQKV
|
7.8 | IC50 | 2 | — | |
CXBBWVXSZINRCS
|
7.8 | Ki | 41 | — | |
TYNGHODBFDMDKR
|
7.8 | IC50 | 3 | — | |
UQJQNZHGEVLHST
|
7.8 | Ki | 15 | — | |
VQPBIJGXSXEOCU
|
7.8 | Ki | 24 | — | |
KXEVSPQLDCBMPG
|
7.7 | IC50 | 2 | — | |
FNZJYDYAQSDVIG
|
7.7 | IC50 | 2 | — | |
FRJOVFNLSNXELB
|
7.7 | IC50 | 3 | — | |
PKUNWOUAVLHPIJ
|
7.7 | IC50 | 2 | — | |
VCHPXQWCAXPYAS
|
7.7 | IC50 | 2 | — | |
JFIZOYQARFPKTF
|
7.7 | IC50 | 2 | — | |
FUZSHLVNKZZEKR
|
7.6 | IC50 | 16 | — | |
KSUDUUBCXJUFRL
|
7.6 | Kd | 12 | — | |
SKDYZXWYDRSLQY
|
7.6 | IC50 | 2 | — | |
RXVAQVGZWRONPW
|
7.6 | IC50 | 2 | — | |
CZQVOIDVDAVDFW
|
7.5 | Ki | 18 | — | |
RNOAOAWBMHREKO
|
7.5 | IC50 | 15 | — | |
UXHHASKNWWRBLI
|
7.5 | IC50 | 3 | — | |
IXGIDKKCSASRGG
|
7.5 | IC50 | 2 | — | |
MREXTQDSRCXTPN
|
7.5 | IC50 | 2 | — | |
SKDSRJRRAQLUPP
|
7.5 | IC50 | 8 | Yes | |
QQWUGDVOUVUTOY
|
7.4 | Kd | 231 | Yes | |
KOLMPPLMZOKCEL
|
7.4 | IC50 | 3 | — | |
SRSQULBCTWSVKL
|
7.4 | IC50 | 15 | — | |
CXQHYVUVSFXTMY
|
7.4 | Kd | 154 | — | |
JDWRBLXGJZCOBR
|
7.4 | IC50 | 2 | — | |
AXMMFQYWZDPEFR
|
7.3 | IC50 | 2 | — |