Target Details
| UniProt AC | Q13873 |
|---|---|
| Gene Symbol | BMPR2 |
| Protein Name | Bone morphogenetic protein receptor type-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF00069 (Pkinase) |
Summary
- Multi-target molecules 26
- Clinical molecules 9
- Avg pChEMBL 6.88
KEGG Pathways (7)
Associated Diseases (3)
Active Molecules (26)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AQSSMEORRLJZLU
|
8.5 | Kd | 34 | Yes | |
RYYNGWLOYLRZLK
|
8.1 | Kd | 45 | — | |
MWKSRKSEWLRPBL
|
7.8 | Kd | 1075 | — | |
WCDLCPLAAKUJNY
|
7.8 | IC50 | 8 | — | |
NHFDRBXTEDBWCZ
|
7.7 | Kd | 12 | Yes | |
IIYOBXCNRFSCBH
|
7.6 | IC50 | 8 | — | |
LOLPPWBBNUVNQZ
|
7.4 | Kd | 97 | Yes | |
XZXHXSATPCNXJR
|
7.2 | Kd | 165 | Yes | |
WMTXIPYJYDISKM
|
7.2 | IC50 | 8 | — | |
XHBVYDAKJHETMP
|
7.1 | IC50 | 24 | Yes | |
YRRRHSNOXWKVDL
|
7.1 | IC50 | 5 | — | |
MFAQYJIYDMLAIM
|
7.0 | Kd | 130 | Yes | |
XLSYZSRXVVCHLS
|
6.8 | Kd | 48 | — | |
BZZKEPGENYLQSC
|
6.7 | IC50 | 6 | — | |
CTNPALGJUAXMMC
|
6.7 | Kd | 151 | — | |
GUBJNPWVIUFSTR
|
6.5 | Kd | 103 | — | |
YYLKKYCXAOBSRM
|
6.4 | Kd | 191 | — | |
OEZHSZIDGUKBRK
|
6.3 | IC50 | 10 | — | |
UBPYILGKFZZVDX
|
6.2 | Kd | 130 | Yes | |
WINHZLLDWRZWRT
|
6.2 | Kd | 201 | Yes | |
BBDGBGOVJPEFBT
|
6.2 | IC50 | 6 | — | |
KDKUVYLMPJIGKA
|
6.1 | Kd | 91 | Yes | |
HFNKQEVNSGCOJV
|
6.0 | Kd | 65 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |