Target Details
| UniProt AC | Q13822 |
|---|---|
| Gene Symbol | ENPP2 |
| Protein Name | Autotaxin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01223 (Endonuclease_NS) PF01663 (Phosphodiest) PF01033 (Somatomedin_B) |
Summary
- Multi-target molecules 261
- Clinical molecules 0
- Avg pChEMBL 7.85
KEGG Pathways (2)
Active Molecules (261)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VKGKTWSBQKAVNC
|
7.4 | IC50 | 2 | — | |
CQATZYOPEZUCOU
|
7.4 | IC50 | 2 | — | |
VXDVTTQURJJEAI
|
7.4 | IC50 | 2 | — | |
WXEFNHJXTXKSAR
|
7.4 | IC50 | 2 | — | |
JNCFYDWBXFRFNI
|
7.4 | IC50 | 2 | — | |
ZKCDXPLZDIFJFJ
|
7.4 | IC50 | 2 | — | |
KJIYUARBMWVZFP
|
7.3 | IC50 | 2 | — | |
ZQXSDNMNMANIPW
|
7.3 | IC50 | 2 | — | |
WUFPYBVDYIRBPK
|
7.3 | IC50 | 2 | — | |
MJSJFHWVIMXAHX
|
7.2 | IC50 | 2 | — | |
DBPDXQVNPSOVIS
|
7.2 | IC50 | 2 | — | |
MYBWJHNUYIIVMQ
|
7.2 | IC50 | 2 | — | |
IZTQHCHOUPBCOP
|
7.2 | IC50 | 2 | — | |
KXVQTJOSXSHGSM
|
7.2 | IC50 | 2 | — | |
QPCFJOICHYLCTB
|
7.2 | IC50 | 2 | — | |
QDRPGHYUNDWJIU
|
7.2 | IC50 | 2 | — | |
ZXSODDRRFJTXOA
|
7.2 | IC50 | 2 | — | |
YWJYAUHBIGXRKD
|
7.1 | IC50 | 2 | — | |
IGKPGOAZPNQIRH
|
7.1 | IC50 | 2 | — | |
IRCLLBJQKIMLIN
|
7.1 | IC50 | 2 | — | |
BEERJOYNULAZMS
|
7.0 | IC50 | 2 | — | |
SRNMGIFMQYRFTQ
|
7.0 | IC50 | 2 | — | |
ZVAPUQBYQNLXGP
|
7.0 | IC50 | 2 | — | |
JUQSJACIWQDEDP
|
7.0 | IC50 | 2 | — | |
SFWJESQUECBVOV
|
7.0 | IC50 | 2 | — | |
MIWTUCTXRDTYFF
|
6.9 | IC50 | 2 | — | |
OTANRZOABZEFKX
|
6.9 | IC50 | 2 | — | |
FKWXMWXKDVIGSP
|
6.9 | IC50 | 2 | — | |
IJYANMWQCFERTA
|
6.9 | IC50 | 2 | — | |
NSVAQEHOXWOGFX
|
6.9 | IC50 | 2 | — | |
IIGWORAYWRDOLY
|
6.9 | IC50 | 2 | — | |
HYIQTVPHAUHFPI
|
6.8 | IC50 | 2 | — | |
XHBMWGNALFPNJS
|
6.8 | IC50 | 2 | — | |
QSDZSKSAPMAMLJ
|
6.8 | IC50 | 2 | — | |
WRGWNNDUOFUGIS
|
6.8 | IC50 | 2 | — | |
YZFIDZNZVKFQOO
|
6.8 | IC50 | 2 | — | |
LMTIYKNLPQQREE
|
6.7 | IC50 | 2 | — | |
UHEJWZYXFUKRNS
|
6.6 | IC50 | 2 | — | |
RDMIFINBVKZJSN
|
6.6 | IC50 | 2 | — | |
UEEMHDQTRLSWSV
|
6.6 | IC50 | 2 | — | |
GIMIOPSJDCYEST
|
6.6 | IC50 | 2 | — | |
CKGFBLVIEYVQDY
|
6.5 | IC50 | 2 | — | |
GEGDEOMKGFQOPG
|
6.5 | IC50 | 2 | — | |
ZUVJKJYJTFBRTK
|
6.5 | IC50 | 2 | — | |
LLVQORFQCYMTJK
|
6.5 | IC50 | 2 | — | |
TWZGGFPYNFZHRE
|
6.5 | IC50 | 2 | — | |
OZEOFYOYWSWOOH
|
6.4 | IC50 | 2 | — | |
COSPWWJGDNPZSN
|
6.4 | IC50 | 2 | — | |
CGZVZUYWLUAMAL
|
6.4 | IC50 | 2 | — | |
WRGQSWVCFNIUNZ
|
6.4 | IC50 | 3 | — |