Target Details
| UniProt AC | Q13822 |
|---|---|
| Gene Symbol | ENPP2 |
| Protein Name | Autotaxin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01223 (Endonuclease_NS) PF01663 (Phosphodiest) PF01033 (Somatomedin_B) |
Summary
- Multi-target molecules 261
- Clinical molecules 0
- Avg pChEMBL 7.85
KEGG Pathways (2)
Active Molecules (261)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JLJPPAFQJMGWJP
|
7.8 | IC50 | 2 | — | |
YMCWUEVNKWTDOD
|
7.8 | IC50 | 2 | — | |
SDAXSYKZYIDSSA
|
7.8 | IC50 | 2 | — | |
OQPVHCISWVIMLV
|
7.8 | IC50 | 2 | — | |
DKWNFDILVIWZNB
|
7.8 | IC50 | 2 | — | |
DPDXALVQOXCYKF
|
7.8 | IC50 | 2 | — | |
FMWQENMZFHAGIB
|
7.8 | IC50 | 2 | — | |
OIVNVRWGAPTUBT
|
7.8 | IC50 | 2 | — | |
AJEXTHORZPSOBR
|
7.8 | IC50 | 2 | — | |
VCHVRSPQMBHYNT
|
7.8 | IC50 | 2 | — | |
DLMICULGTDCPSM
|
7.8 | IC50 | 2 | — | |
DAIJYTRDFYRRPE
|
7.8 | IC50 | 2 | — | |
IFXXYODLELYUIJ
|
7.8 | IC50 | 2 | — | |
NQTQJEQNOKRCLR
|
7.8 | IC50 | 2 | — | |
OPTARTWTKNYZKR
|
7.8 | IC50 | 2 | — | |
QUWQVGMGYNONEZ
|
7.8 | IC50 | 2 | — | |
DYNFMEUREYYYSN
|
7.8 | IC50 | 2 | — | |
AZFLZKYAFIGXSQ
|
7.7 | IC50 | 2 | — | |
KGLFVEGJSIFVRF
|
7.7 | IC50 | 2 | — | |
QQGIJLAOOUAFTR
|
7.7 | IC50 | 2 | — | |
UYSQGHYYHXJDTD
|
7.7 | IC50 | 2 | — | |
IFDFEOVSVMPHCS
|
7.7 | IC50 | 2 | — | |
PFYGFLKRYKKYEU
|
7.7 | IC50 | 2 | — | |
RZDILIUVLNUMGK
|
7.7 | IC50 | 2 | — | |
YMILTOKXDKHMQW
|
7.7 | IC50 | 2 | — | |
IZQVHGHBYZROSX
|
7.7 | IC50 | 2 | — | |
IFDFEOVSVMPHCS
|
7.7 | IC50 | 2 | — | |
VAWHLBLARXWUKL
|
7.7 | IC50 | 2 | — | |
KETUZQKXCLKERW
|
7.7 | IC50 | 2 | — | |
SFMXRLAXDHNNBZ
|
7.7 | IC50 | 2 | — | |
LOMCGZAQBNLPJR
|
7.7 | IC50 | 2 | — | |
XCGGPJPPGDCVNV
|
7.7 | IC50 | 2 | — | |
OPMLSLQOQSGBDC
|
7.6 | IC50 | 2 | — | |
XHZBBSUUPYBQGC
|
7.6 | IC50 | 2 | — | |
QZEJPCSNGFLHEW
|
7.6 | IC50 | 2 | — | |
WZBWCZRXSCQZSZ
|
7.6 | IC50 | 2 | — | |
QYGGUPLMEGCJJA
|
7.6 | IC50 | 2 | — | |
ZTCPZDCGSZMOPQ
|
7.6 | IC50 | 2 | — | |
CHMCNIRNOVQGFL
|
7.6 | IC50 | 2 | — | |
FDWYOSZDAODUPT
|
7.6 | IC50 | 2 | — | |
MHRZSBMHABOVDN
|
7.6 | IC50 | 2 | — | |
GORMEHYDOGSCDJ
|
7.6 | IC50 | 2 | — | |
NLAXMHQWTOCNAO
|
7.5 | IC50 | 3 | — | |
YYJNDZDFZZFANH
|
7.5 | IC50 | 2 | — | |
BWCSDDAQCDQZFW
|
7.5 | IC50 | 2 | — | |
LLKASGYDVIKVNO
|
7.5 | IC50 | 2 | — | |
VMOAEQWYVOQCMP
|
7.4 | IC50 | 2 | — | |
SAUMRYSIRCXBFC
|
7.4 | IC50 | 2 | — | |
RSUYEIKCLHSVRW
|
7.4 | IC50 | 2 | — | |
TYXSCUWWRHCFPA
|
7.4 | IC50 | 2 | — |