Target Details
| UniProt AC | Q13822 |
|---|---|
| Gene Symbol | ENPP2 |
| Protein Name | Autotaxin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01223 (Endonuclease_NS) PF01663 (Phosphodiest) PF01033 (Somatomedin_B) |
Summary
- Multi-target molecules 261
- Clinical molecules 0
- Avg pChEMBL 7.85
KEGG Pathways (2)
Active Molecules (261)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YMNUUEPTOAODOJ
|
8.1 | IC50 | 2 | — | |
ZVQCTFSUZGCCIM
|
8.1 | IC50 | 2 | — | |
DSWPTVKCBCROGK
|
8.1 | IC50 | 3 | — | |
AASOGRFONRFNKH
|
8.1 | IC50 | 2 | — | |
HOLGWONGFZVVTN
|
8.1 | IC50 | 2 | — | |
LUOJVXWFMUOXAE
|
8.1 | IC50 | 2 | — | |
MPJUJKDYBYAOAV
|
8.1 | IC50 | 2 | — | |
RDQNCXQQDOPWRG
|
8.1 | IC50 | 2 | — | |
SATKYBKQMZMOTQ
|
8.1 | IC50 | 2 | — | |
SGVMFTNWXPQKEJ
|
8.1 | IC50 | 2 | — | |
TXRSJAFBRCLJBE
|
8.1 | IC50 | 2 | — | |
VNOABWFAQZFZOI
|
8.1 | IC50 | 2 | — | |
VOPKNELFOUYEOQ
|
8.1 | IC50 | 2 | — | |
YLIKCNACGAJJCL
|
8.1 | IC50 | 2 | — | |
ZVAPUQBYQNLXGP
|
8.1 | IC50 | 2 | — | |
ACTRSKZFXVVKJF
|
8.0 | IC50 | 2 | — | |
DSLJISHBSCLIEH
|
8.0 | IC50 | 2 | — | |
FAAGHBOJELRUFX
|
8.0 | IC50 | 2 | — | |
GQIYQQWGUUFVAK
|
8.0 | IC50 | 2 | — | |
IHNCKMJGCJAJDW
|
8.0 | IC50 | 2 | — | |
JFLVMQRHUVHYBM
|
8.0 | IC50 | 2 | — | |
JMWIYCDNOVTMIF
|
8.0 | IC50 | 2 | — | |
MFAFPFCSTKBXTH
|
8.0 | IC50 | 2 | — | |
NQACASOSTXVQFQ
|
8.0 | IC50 | 2 | — | |
PEXIQROTQWLYBW
|
8.0 | IC50 | 2 | — | |
PMMLAGCGRWXTKW
|
8.0 | IC50 | 2 | — | |
SKNHHIBJRMDTNP
|
8.0 | IC50 | 2 | — | |
UOACMELVYDGMSF
|
8.0 | IC50 | 2 | — | |
UZTXHXYLFOLAIC
|
8.0 | IC50 | 2 | — | |
XPUKIZYEZJYAFE
|
8.0 | IC50 | 2 | — | |
YWJYAUHBIGXRKD
|
8.0 | IC50 | 2 | — | |
XHLDHHAKCKRBKN
|
8.0 | IC50 | 2 | — | |
PMYVQHJLSGSLJR
|
8.0 | IC50 | 2 | — | |
DDVSVIYUNGBPCE
|
8.0 | IC50 | 2 | — | |
DYMPGPPORQYWQU
|
8.0 | IC50 | 2 | — | |
KYTPMRUGEHJYJI
|
8.0 | IC50 | 2 | — | |
MEZDYULALVWYSZ
|
8.0 | IC50 | 2 | — | |
YBUPNURAXMMCKO
|
8.0 | IC50 | 2 | — | |
CRBIPFHCBLHMGJ
|
7.9 | IC50 | 2 | — | |
AQXAJKJTOQIJCR
|
7.9 | IC50 | 2 | — | |
GTOOLRZGLJZZBK
|
7.9 | IC50 | 2 | — | |
XGHTXOLGJNRNKS
|
7.9 | IC50 | 2 | — | |
HEWIQRKZRSQSHI
|
7.9 | IC50 | 2 | — | |
LFXSEFMFDJZNPP
|
7.9 | IC50 | 2 | — | |
MNESUNURENQFHQ
|
7.9 | IC50 | 2 | — | |
UIZIAVWJJSSOCV
|
7.9 | IC50 | 2 | — | |
UTICIZWBNOHDIF
|
7.9 | IC50 | 2 | — | |
VSTOHOUVPQCSIT
|
7.9 | IC50 | 2 | — | |
SIBYCEPFLIGWEY
|
7.9 | IC50 | 2 | — | |
GDBSDPMVPGTXNU
|
7.8 | IC50 | 2 | — |