Target Details
| UniProt AC | Q13822 |
|---|---|
| Gene Symbol | ENPP2 |
| Protein Name | Autotaxin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01223 (Endonuclease_NS) PF01663 (Phosphodiest) PF01033 (Somatomedin_B) |
Summary
- Multi-target molecules 261
- Clinical molecules 0
- Avg pChEMBL 7.85
KEGG Pathways (2)
Active Molecules (261)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AJEXTHORZPSOBR
|
9.0 | IC50 | 2 | — | |
AJEXTHORZPSOBR
|
9.0 | IC50 | 2 | — | |
BUPCUEOCEWPZKQ
|
9.0 | IC50 | 2 | — | |
CCYQBVTYCWKICH
|
9.0 | IC50 | 2 | — | |
FMFIJGUAEGKLNT
|
9.0 | IC50 | 2 | — | |
IEQOUKRLORXTRH
|
9.0 | IC50 | 2 | — | |
IHDSOHZJFSYDSW
|
9.0 | IC50 | 2 | — | |
KJTSUDNAUXPLHU
|
9.0 | IC50 | 2 | — | |
LRBMHEFLWCPAKK
|
9.0 | IC50 | 2 | — | |
NDONGBDLTYRPQB
|
9.0 | IC50 | 2 | — | |
PKAFZJIZJFKXPG
|
9.0 | IC50 | 2 | — | |
PZASAAIJIFDWSB
|
9.0 | IC50 | 2 | — | |
REHYZYIYLUIPNH
|
9.0 | IC50 | 2 | — | |
SHYCEMRGCOHMPN
|
9.0 | IC50 | 2 | — | |
VUHNBQOHNTYKHV
|
9.0 | IC50 | 2 | — | |
YHIBNXMKXSVXAN
|
9.0 | IC50 | 2 | — | |
YIKJMTFIKWVVDM
|
9.0 | IC50 | 2 | — | |
YIPRECKELCXDLC
|
9.0 | IC50 | 2 | — | |
YMDDSFMLTGLUOI
|
9.0 | IC50 | 2 | — | |
ZCIQNLYHYPYKMT
|
9.0 | IC50 | 2 | — | |
ZVAPUQBYQNLXGP
|
9.0 | IC50 | 2 | — | |
ZVIDGTNRDBKHRC
|
9.0 | IC50 | 2 | — | |
YNNILJZFEPDRJM
|
8.9 | IC50 | 2 | — | |
GFGRUPJITXXZQN
|
8.7 | IC50 | 2 | — | |
AZFNTAYQQKHJRM
|
8.7 | IC50 | 2 | — | |
IOLORNUXBZHBTP
|
8.7 | IC50 | 2 | — | |
JIGKNSVZQIRWLK
|
8.7 | IC50 | 2 | — | |
LPFFWGOZXIUBKT
|
8.7 | IC50 | 2 | — | |
QIENJTFBCLUNOG
|
8.7 | IC50 | 2 | — | |
VNBBIBZHRDGYMA
|
8.7 | IC50 | 2 | — | |
WBQHVXBARQTRQI
|
8.7 | IC50 | 2 | — | |
GQDFANKSIDIEMO
|
8.6 | IC50 | 2 | — | |
BIGVDRATVPAKAS
|
8.6 | IC50 | 2 | — | |
HFJGRHYPTCNSKW
|
8.6 | IC50 | 2 | — | |
OGDGBLWCOWZVFO
|
8.6 | IC50 | 2 | — | |
BVQNNVPVXUMBJN
|
8.5 | IC50 | 2 | — | |
DKGWFJXODFKPJZ
|
8.5 | IC50 | 2 | — | |
JMSUDQYHPSNBSN
|
8.5 | IC50 | 2 | — | |
KZXRDHBMXSDWDX
|
8.5 | IC50 | 2 | — | |
LZXUVWUXKWKZOC
|
8.5 | IC50 | 2 | — | |
WYFPTWWEAHNRRX
|
8.5 | IC50 | 2 | — | |
XSPZRFRUMUKODI
|
8.5 | IC50 | 2 | — | |
YMCWUEVNKWTDOD
|
8.5 | IC50 | 2 | — | |
ZRYCTQBOQQJWNH
|
8.5 | IC50 | 2 | — | |
FEUNHRLAPAPVII
|
8.4 | IC50 | 2 | — | |
KZWCVIBEUNXBPZ
|
8.4 | IC50 | 2 | — | |
DFDVFDLIWVLQIA
|
8.4 | IC50 | 2 | — | |
FMZIUIFYMJWAEE
|
8.4 | IC50 | 2 | — | |
GJWHUAAMXSTOQC
|
8.4 | IC50 | 2 | — | |
GPRRGWBAPIJEBL
|
8.4 | IC50 | 2 | — |