Target Details
| UniProt AC | Q13705 |
|---|---|
| Gene Symbol | ACVR2B |
| Protein Name | Activin receptor type-2B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF00069 (Pkinase) |
Summary
- Multi-target molecules 12
- Clinical molecules 3
- Avg pChEMBL 7.19
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (12)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MWKSRKSEWLRPBL
|
8.5 | Kd | 1075 | — | |
MFAQYJIYDMLAIM
|
8.1 | Kd | 130 | Yes | |
VAARYSWULJUGST
|
8.0 | Kd | 119 | Yes | |
KJUCPVIVNLPLEE
|
8.0 | IC50 | 10 | — | |
FHTCHCUICJOIGJ
|
7.8 | IC50 | 7 | — | |
YOKGFEAEVZNOAR
|
7.2 | IC50 | 5 | — | |
FYSRKRZDBHOFAY
|
7.0 | Kd | 8 | — | |
IAYGCINLNONXHY
|
6.6 | Kd | 50 | — | |
YYLKKYCXAOBSRM
|
6.4 | Kd | 191 | — | |
JMGXJHWTVBGOKG
|
6.4 | Kd | 7 | — | |
ZBNZXTGUTAYRHI
|
6.2 | Kd | 102 | Yes | |
JUUFLLKHNYWHKP
|
6.0 | Kd | 12 | — |