Target Details
| UniProt AC | Q13639 |
|---|---|
| Gene Symbol | HTR4 |
| Protein Name | 5-hydroxytryptamine receptor 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 85
- Clinical molecules 1
- Avg pChEMBL 7.93
KEGG Pathways (5)
Active Molecules (85)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JWNWVBYZLJCIIB
|
7.4 | Ki | 3 | — | |
DUUYHLUSDHATNS
|
7.4 | Ki | 3 | — | |
AEHUGLUJLXQXMZ
|
7.3 | Ki | 2 | — | |
MZRKHUUDDHJVHS
|
7.3 | Ki | 2 | — | |
NAPNJRUKMMPNCH
|
7.3 | Ki | 2 | — | |
DZXRSFAKIAKMMD
|
7.3 | Ki | 2 | — | |
OKFGYYBZAZENKT
|
7.2 | Ki | 2 | — | |
DCSUBABJRXZOMT
|
7.2 | Ki | 24 | — | |
OBSQXMOZMFTQSH
|
7.2 | Ki | 2 | — | |
VDFVGSSOSOLGGL
|
7.2 | Ki | 2 | — | |
TXCGMRVPXUBHAL
|
7.1 | Ki | 2 | — | |
ZSTKHSQDNIGFLM
|
7.1 | Kd | 22 | — | |
OTIIXGVFBWDUDH
|
7.0 | Ki | 2 | — | |
DCSUBABJRXZOMT
|
7.0 | Ki | 2 | — | |
GZDHJUWAZOBOGE
|
6.9 | Ki | 2 | — | |
PCGROECTIBEWPF
|
6.9 | Ki | 2 | — | |
UHGWCPXBDDWAKP
|
6.9 | Ki | 2 | — | |
XEHQZRKZBJQOMJ
|
6.9 | Ki | 2 | — | |
BXNNACCQTQBSOO
|
6.8 | Ki | 3 | — | |
YPELFRMCRYSPKZ
|
6.8 | Ki | 9 | — | |
CPQKZLNBCUOHCW
|
6.8 | Ki | 3 | — | |
DAQIUCFPMNHHQR
|
6.7 | Ki | 2 | — | |
ZNRGQMMCGHDTEI
|
6.7 | Ki | 9 | — | |
DUQKAXNRVJCRQH
|
6.7 | Ki | 4 | — | |
QZAYGJVTTNCVMB
|
6.6 | Ki | 17 | — | |
FEROPKNOYKURCJ
|
6.5 | Ki | 8 | — | |
WMCLJWPYJWRZJT
|
6.4 | Ki | 5 | — | |
JTEJPPKMYBDEMY
|
6.4 | Ki | 9 | — | |
VRBLZQPTWBRDKL
|
6.3 | Ki | 3 | — | |
WBYHTZYHAFNBKW
|
6.3 | Ki | 5 | — | |
SPRYLBSGZYATLJ
|
6.2 | Ki | 3 | — | |
BOHGZALGHLQJNA
|
6.1 | IC50 | 7 | — | |
CZWRMNRSJXHJBY
|
6.0 | Ki | 3 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — | |
YOGJZQGRTVMCPY
|
6.0 | IC50 | 17 | — |