Target Details
UniProt ACQ13639
Gene SymbolHTR4
Protein Name5-hydroxytryptamine receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 85
  • Clinical molecules 1
  • Avg pChEMBL 7.93
Top Co-occurrence Targets
Active Molecules (85)
InChIKey pChEMBL Type Targets Clinical
UVOCSZKGWJOKNN 12.2 Ki 11
JBPBJYKHTQKMKP 10.4 Ki 4
AOOSJYIINXVNHV 10.2 Ki 16
KIIQBPBFXXBVSD 10.1 Ki 2
FPDZVPWWAWOFQS 10.0 Ki 2
RNXYMZNGMNWKMC 10.0 Ki 3
RVXJKDQROPYYOF 10.0 Ki 2
OPCCXGXGEHABFP 9.8 Kd 17
YKBQHBXRXWGQIZ 9.7 Ki 3
GDRLBCZDGQFDCZ 9.6 Ki 7
MOZPSIXKYJUTKI 9.6 Ki 2
SMPAXQNASQVLJD 9.6 Ki 2
BIAZRDQNRJRCRQ 9.6 Ki 2
BCGWQEUPMDMJNV 9.0 IC50 30 Yes
UWMNAFXETUEZJZ 8.9 Ki 4
FWCCAIJRQHYBFE 8.9 Ki 2
UVEYNCQCHBIENE 8.8 Ki 2
FJLWRVJMCXVJOE 8.7 Ki 2
WKWADEWWLCVVLF 8.7 Ki 14
YJAIZWWQRYKSON 8.7 Ki 2
WLHFUBIRAHRPHA 8.7 Ki 5
DZZIAERGLDKTBT 8.6 Ki 2
RUCWXMRMXGLFKN 8.6 Ki 2
RYDDBILRWHKYGG 8.6 Ki 2
RVKSBAURRKECBI 8.5 Ki 2
VUPLWNSHTPTZLS 8.5 Ki 2
KMWRABRPTOODHP 8.5 Ki 4
PXUUPGSNIMQISW 8.4 Ki 2
YVCAJCVHBUZCNX 8.4 Ki 2
IKBKZGMPCYNSLU 8.4 Ki 13
GGQFEMQQQLOYIH 8.3 Ki 3
FFNWMBDISAYHDC 8.2 Ki 2
MREMSPSMZSVSJS 8.1 Ki 3
FSZQXBYUVRKUIV 8.1 Ki 2
HBJRTZJDKYEAKF 8.1 Ki 2
YKSIZFAAHBYGMG 8.1 Ki 2
UOOCXIPKYHHRRD 8.1 Ki 2
JBHLYIVFFLNISJ 8.0 Ki 2
FTRZTHFGTILUPE 8.0 Ki 3
KVVCXQIQAOOKFF 8.0 Ki 3
BFZKHVUFJAQCQW 7.9 Ki 2
ZAKCOJKXWMIQSX 7.9 Ki 2
DHFMNRHFVSQCPD 7.8 Ki 2
LZSQXRQOXNBANQ 7.8 Ki 2
OLINRUQQUFMPJJ 7.8 Ki 2
QPDCBQORMYFXGT 7.8 Ki 2
HISLDJKGFNEVLO 7.7 Ki 2
MIVZTSHUBPAZML 7.7 Ki 3
MIGORCBCNUSMCM 7.6 Ki 2
JBJVWRHVBXWURS 7.4 Ki 2
2D structure