Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MFLKPCAUPXBTPC
|
7.4 | IC50 | 5 | — | |
MNPDDWGYJIGNTR
|
7.4 | IC50 | 2 | — | |
QCTMVDQWYGRUJK
|
7.4 | IC50 | 9 | — | |
VJSOYRZFTRFBFM
|
7.4 | IC50 | 5 | — | |
ACOQCSBMVFAWQV
|
7.3 | IC50 | 8 | — | |
LVSVYVPFNYRNOF
|
7.3 | IC50 | 8 | — | |
FKRHOHUJMCOWDZ
|
7.3 | IC50 | 5 | — | |
IMSFHJBONZQKCR
|
7.3 | IC50 | 2 | — | |
QCHDHJOEPUQALZ
|
7.3 | IC50 | 9 | — | |
YDTHCIZMSQZYMR
|
7.3 | IC50 | 9 | — | |
FSICBNKCBMOCOY
|
7.3 | IC50 | 2 | — | |
RUQXGVGYNKIGJD
|
7.3 | IC50 | 6 | — | |
ZUADZDBGZDSSAB
|
7.3 | IC50 | 5 | — | |
BXNJHAXVSOCGBA
|
7.3 | IC50 | 14 | — | |
CIGFCAJNHRIRIV
|
7.3 | IC50 | 2 | — | |
KQCIEIGKPXQRLM
|
7.3 | IC50 | 6 | — | |
ADJWQFUAOONPHD
|
7.3 | IC50 | 8 | — | |
CHADTINFLWZSKR
|
7.3 | Ki | 26 | — | |
DCPBIOSSTDLFHO
|
7.3 | IC50 | 3 | — | |
FFESRGFMLQEDRD
|
7.3 | IC50 | 5 | — | |
HJYHJYGXRBYDIG
|
7.3 | Ki | 23 | — | |
KOHNRDPXFDZZJF
|
7.3 | Ki | 31 | — | |
LACOMQAWPSFXQC
|
7.3 | Ki | 27 | — | |
LOCWELCIOZHZHE
|
7.3 | Ki | 11 | — | |
LZUJDIWVWSRLRQ
|
7.3 | IC50 | 4 | — | |
LZUJDIWVWSRLRQ
|
7.3 | IC50 | 4 | — | |
MVJMMLFMPWITEJ
|
7.3 | Ki | 110 | — | |
NBIWQDNWQHQXFS
|
7.3 | IC50 | 5 | — | |
OUJZYQBEFNDJQN
|
7.3 | Ki | 71 | — | |
RGOPHVZLEMGMBZ
|
7.3 | Ki | 20 | — | |
SZOYOCHRMSEEMG
|
7.3 | IC50 | 3 | — | |
TWCARTFPHQNBPF
|
7.3 | Ki | 16 | — | |
UMYSGMXAOXMMGG
|
7.3 | IC50 | 7 | — | |
XTJRKTBELWGSDN
|
7.3 | IC50 | 8 | — | |
YGUMGYOBTNGZKS
|
7.3 | Ki | 12 | — | |
PAEFKCSDRFLRMD
|
7.3 | IC50 | 5 | — | |
RUQXGVGYNKIGJD
|
7.3 | IC50 | 7 | — | |
ASLGQVPNOSGBQR
|
7.3 | IC50 | 10 | — | |
DDLZLOKCJHBUHD
|
7.3 | IC50 | 23 | — | |
FPFBUUBVECCCFK
|
7.3 | IC50 | 2 | — | |
JGJABYQWCCWLPP
|
7.3 | IC50 | 4 | — | |
JXQZHHAAJMQJKU
|
7.3 | IC50 | 6 | — | |
CXJCGSPAPOTTSF
|
7.3 | IC50 | 3 | — | |
CXJCGSPAPOTTSF
|
7.3 | IC50 | 6 | — | |
BZNZVNQDMRWLSV
|
7.2 | IC50 | 2 | — | |
CRLFBJGERQILPV
|
7.2 | Ki | 2 | — | |
IDOKKOQIQLHASZ
|
7.2 | IC50 | 8 | — | |
KOMXYYABYRRJBD
|
7.2 | IC50 | 3 | — | |
DSCUTYQYWCTFQL
|
7.2 | IC50 | 6 | — | |
OAUMCWJJYNUCIM
|
7.2 | IC50 | 5 | — |