Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OEVQTWCGWDOIFZ
|
7.5 | IC50 | 6 | — | |
WFOMWAYINPJPDX
|
7.5 | IC50 | 9 | — | |
XLSYZSRXVVCHLS
|
7.5 | Kd | 48 | — | |
OTKZKCGOQJKFMT
|
7.5 | IC50 | 4 | — | |
POCZBHBFCIWCCV
|
7.5 | IC50 | 5 | — | |
UKWWUFBDIVBOBD
|
7.5 | IC50 | 5 | — | |
VPLSDHGYIYFKRM
|
7.5 | IC50 | 2 | — | |
WKYMGORXOQPTTO
|
7.5 | IC50 | 9 | — | |
WQYUNADCLFWKGN
|
7.5 | IC50 | 7 | — | |
JLGZOWVGNXABBW
|
7.4 | Ki | 2 | — | |
PPZINUUIYSVIGC
|
7.4 | IC50 | 6 | — | |
CEDLXWRFEZCVEU
|
7.4 | IC50 | 2 | — | |
PPQSZAVBAJMLRF
|
7.4 | IC50 | 5 | — | |
YBASBPWQGVPOIX
|
7.4 | IC50 | 2 | — | |
KBEZZFIQPRMPRG
|
7.4 | IC50 | 5 | — | |
LIYXXFOSHNQSRD
|
7.4 | IC50 | 4 | Yes | |
VOXHNNQHNDOGSK
|
7.4 | IC50 | 4 | — | |
JWICEQLMDWKZGQ
|
7.4 | IC50 | 2 | — | |
LLMXWBSEQIDLJG
|
7.4 | IC50 | 5 | — | |
OCVVFPATGNRPNO
|
7.4 | IC50 | 2 | — | |
YGXHQYJKJUFSJI
|
7.4 | IC50 | 14 | — | |
AOBLBPWPSKBHSI
|
7.4 | Ki | 55 | — | |
FAIHBCXQSBIRIL
|
7.4 | Ki | 22 | — | |
GVMDVMPNOAVKJR
|
7.4 | Ki | 26 | Yes | |
HNODKCFEFLQKBO
|
7.4 | Ki | 6 | — | |
HOYRWTWZUFFACV
|
7.4 | Ki | 28 | — | |
HXESDBWWDYJEJQ
|
7.4 | Ki | 10 | — | |
JANQPHRPUAYQTA
|
7.4 | IC50 | 5 | — | |
JJWLXRKVUJDJKG
|
7.4 | Kd | 6 | — | |
JLTBOCSFMNSLFH
|
7.4 | Ki | 9 | — | |
KCKXYZOBGBJZEG
|
7.4 | Ki | 36 | — | |
NLUPJKQOKWBWFC
|
7.4 | Ki | 69 | — | |
PLHUMPJXRHMFFR
|
7.4 | Ki | 28 | — | |
QCLXNOBXQUWUEW
|
7.4 | IC50 | 9 | — | |
SGHXFHRRWFLILP
|
7.4 | Ki | 29 | — | |
UCULOFHOCATNHB
|
7.4 | IC50 | 2 | — | |
UZFPGFONVYFSRR
|
7.4 | Ki | 16 | — | |
VQAZMVUNBILJGW
|
7.4 | IC50 | 5 | — | |
XUFLBSMTYMFOQH
|
7.4 | Ki | 43 | — | |
LJQLTQRHIJBENP
|
7.4 | IC50 | 2 | — | |
PCIQNDJCGPAWGK
|
7.4 | IC50 | 2 | — | |
TUIPZIRQUAZXFN
|
7.4 | IC50 | 2 | — | |
VCFPJHJKTXRDGD
|
7.4 | IC50 | 3 | — | |
BWORFRWIDWQHPL
|
7.4 | IC50 | 7 | — | |
HPYSMRPYCUVINY
|
7.4 | IC50 | 2 | — | |
NNPWUWSWEGWPMQ
|
7.4 | IC50 | 8 | — | |
ATXGVVQAUKKFAN
|
7.4 | IC50 | 4 | — | |
OJSLNTSFMXRUEG
|
7.4 | IC50 | 2 | — | |
ZSZSXTFUWZNVBW
|
7.4 | IC50 | 2 | — | |
GVQSROMOXGBVJP
|
7.4 | IC50 | 2 | — |