Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QFBOPHGXTBOQRN
|
7.6 | IC50 | 7 | — | |
RILDWXOQLWEXDG
|
7.6 | IC50 | 6 | — | |
UHOPJKMQVDXYAV
|
7.6 | IC50 | 8 | — | |
QDNBLKZVYODRLC
|
7.6 | IC50 | 5 | — | |
MYLYCZDLVLCRLU
|
7.5 | IC50 | 5 | — | |
YSMNHYFBBOMUFX
|
7.5 | Kd | 3 | — | |
ZBYBDKHFLSHGBP
|
7.5 | IC50 | 4 | — | |
ZBYBDKHFLSHGBP
|
7.5 | IC50 | 4 | — | |
ZQZULRTVXPNQNP
|
7.5 | IC50 | 4 | — | |
KCTCLVINURCCIL
|
7.5 | IC50 | 7 | — | |
CCUMIOKJQCVBML
|
7.5 | IC50 | 2 | — | |
FMWMKOOUBGJSJD
|
7.5 | IC50 | 4 | — | |
HAFFBDGNUZMNIJ
|
7.5 | IC50 | 7 | — | |
RQFGUPSBOAVFSQ
|
7.5 | IC50 | 2 | — | |
SOHWYEVCBPDAIO
|
7.5 | IC50 | 3 | — | |
SQWZFLMPDUSYGV
|
7.5 | IC50 | 11 | — | |
SQWZFLMPDUSYGV
|
7.5 | IC50 | 8 | — | |
ABRIIMZXUFHPCH
|
7.5 | IC50 | 5 | — | |
JJUHKRNDDMOYGK
|
7.5 | IC50 | 3 | — | |
LXDHFJUOCGKVAV
|
7.5 | IC50 | 5 | — | |
BEJCLDKQCNVTQR
|
7.5 | Ki | 16 | — | |
CALAEFSQWBJMDU
|
7.5 | Ki | 21 | — | |
CPGKMMMSMJKHDL
|
7.5 | Ki | 16 | — | |
CYLGCMABIBXHIQ
|
7.5 | Ki | 16 | — | |
GCBJDOWIQHMCMR
|
7.5 | Ki | 84 | — | |
IPKHSYHXXAIZDD
|
7.5 | Ki | 18 | — | |
KAICHBSRWFIESE
|
7.5 | Ki | 14 | — | |
KAZJIBCOYQRDGG
|
7.5 | Ki | 16 | — | |
KTWBYGUSEYSRND
|
7.5 | Ki | 28 | — | |
PGPHHJBZEGSUNE
|
7.5 | IC50 | 3 | — | |
RGKOSKZCLZXDJI
|
7.5 | IC50 | 4 | — | |
RRAMBEGOYIJQHY
|
7.5 | Ki | 11 | — | |
RWKDVIAVTRRJIR
|
7.5 | Ki | 23 | — | |
SBFPHSVZEXSHTL
|
7.5 | Ki | 62 | — | |
TWECFLXNJZAZBE
|
7.5 | IC50 | 2 | — | |
URXJBXVGNBGIJA
|
7.5 | IC50 | 9 | — | |
XKBACCJVCIHQMK
|
7.5 | IC50 | 2 | — | |
XSDJOIOVIMPMHD
|
7.5 | Ki | 44 | — | |
YYSXUOHHBBMQMJ
|
7.5 | IC50 | 7 | — | |
ZGDYBJXDIXVTLV
|
7.5 | Ki | 54 | — | |
DGTHPUFVPBPNPD
|
7.5 | IC50 | 3 | — | |
BDWKOEXYKJGIMA
|
7.5 | IC50 | 2 | — | |
COYCDCAUDJBGOV
|
7.5 | IC50 | 6 | — | |
FWFWXUJORMCFKY
|
7.5 | IC50 | 3 | — | |
QXMXIHBLICGPMG
|
7.5 | IC50 | 9 | — | |
RYWACTNAXCMTTN
|
7.5 | IC50 | 9 | — | |
UTDNMHFLZJFPPY
|
7.5 | IC50 | 4 | — | |
XGDCSHCKBNJGMN
|
7.5 | IC50 | 2 | — | |
ATVTUVKVZSYFBE
|
7.5 | IC50 | 7 | — | |
MDPBVLVUPMAUIA
|
7.5 | IC50 | 2 | — |