Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IJFKKIMDRSZOOW
|
7.7 | IC50 | 6 | — | |
PCUWPDUAQBAWHT
|
7.7 | IC50 | 4 | — | |
PGPHHJBZEGSUNE
|
7.7 | IC50 | 4 | — | |
QTRZNDLLYHSJSH
|
7.7 | IC50 | 9 | — | |
RVSKJUNTDGBSSS
|
7.7 | Ki | 25 | — | |
SQXSMLLCDWJNAC
|
7.7 | Ki | 20 | — | |
SRONQUHCRFZABC
|
7.7 | Ki | 28 | — | |
UIARLYUEJFELEN
|
7.7 | Kd | 289 | Yes | |
XTJRKTBELWGSDN
|
7.7 | IC50 | 8 | — | |
CHQYAWLKOUOTQO
|
7.7 | IC50 | 7 | — | |
BYUPNMOFJSAIHN
|
7.7 | IC50 | 6 | — | |
LCSMODPSWXEJLH
|
7.7 | IC50 | 3 | — | |
WFOMWAYINPJPDX
|
7.7 | IC50 | 9 | — | |
YHZQZEGQCKWCLP
|
7.7 | IC50 | 9 | — | |
CQKBSRPVZZLCJE
|
7.7 | IC50 | 2 | — | |
FEZCHKAGMYXVNX
|
7.7 | IC50 | 6 | — | |
VEZMWMSMHXKTFY
|
7.7 | IC50 | 4 | — | |
YMIDGKZVYFXIBW
|
7.7 | IC50 | 8 | — | |
ZBKFRVXDYILXFJ
|
7.7 | IC50 | 6 | — | |
KOEMSQCYTSQEEQ
|
7.7 | IC50 | 2 | — | |
DXVSNYWBRDTHFF
|
7.6 | IC50 | 7 | — | |
JRNJNYBQQYBCLE
|
7.6 | Kd | 40 | Yes | |
LXQXBEIFOYAXOP
|
7.6 | IC50 | 9 | — | |
QXPJTIYARGTANC
|
7.6 | IC50 | 3 | — | |
UZWDCWONPYILKI
|
7.6 | IC50 | 47 | — | |
WXMYTQDKBPDSSR
|
7.6 | IC50 | 4 | — | |
YRFAWSIUIFNVQA
|
7.6 | IC50 | 9 | — | |
BKIAHCJPMJSHSQ
|
7.6 | IC50 | 6 | — | |
KAEULNCNLILYLK
|
7.6 | IC50 | 4 | — | |
PGPHHJBZEGSUNE
|
7.6 | IC50 | 21 | — | |
PGPHHJBZEGSUNE
|
7.6 | IC50 | 17 | — | |
PUGXENIKUPHCAF
|
7.6 | IC50 | 2 | — | |
WCJBJECTLLTBHS
|
7.6 | IC50 | 2 | — | |
BQWACEUCYSZDBQ
|
7.6 | Ki | 5 | — | |
CNQGNADBGYCKKV
|
7.6 | Ki | 25 | — | |
CRKQBJZCCHKEGI
|
7.6 | Ki | 20 | — | |
JOIUJUJSHIHBDT
|
7.6 | Ki | 18 | — | |
ODNOTLMFNVWFTJ
|
7.6 | Ki | 11 | — | |
PCQMERRARZKTPW
|
7.6 | Ki | 68 | — | |
RGNHKJWHFIPHIM
|
7.6 | Ki | 66 | — | |
SKKRZILJUKYLJS
|
7.6 | Ki | 25 | — | |
UVJQEKJPAVSBTA
|
7.6 | IC50 | 8 | — | |
WDARYLSSWBWVCU
|
7.6 | Ki | 49 | — | |
BYMPGMQLSBLSIU
|
7.6 | IC50 | 5 | — | |
FGBSSPMQGRUJPS
|
7.6 | IC50 | 10 | — | |
GDFYUGGDTISZFA
|
7.6 | IC50 | 2 | — | |
KNLSVEADBVICIJ
|
7.6 | IC50 | 5 | — | |
ZWDRSWWQYGLOOM
|
7.6 | IC50 | 2 | — | |
AQDWDWAYVBQMAM
|
7.6 | IC50 | 7 | — | |
MQRHLOPPMRFMKM
|
7.6 | IC50 | 9 | — |