Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KRWCFCQJKXIENS
|
7.9 | IC50 | 3 | — | |
FFJGYBJUQCZAAY
|
7.8 | IC50 | 5 | — | |
IJFKKIMDRSZOOW
|
7.8 | IC50 | 9 | — | |
UUIPRATXTHJYHH
|
7.8 | IC50 | 3 | — | |
WREJZZXSNOJGIW
|
7.8 | IC50 | 9 | — | |
GLCIBEGENZSGCS
|
7.8 | IC50 | 3 | — | |
MLAPBLMPGXKRBF
|
7.8 | IC50 | 3 | — | |
POSGRZQCKOTBHE
|
7.8 | IC50 | 3 | — | |
ANKYADWZYKSCAJ
|
7.8 | IC50 | 7 | — | |
DJHMDVUOYUYLOJ
|
7.8 | IC50 | 9 | — | |
JHKYWRMDSIQKSV
|
7.8 | IC50 | 2 | — | |
LGUYVFVZZRHOGY
|
7.8 | IC50 | 2 | — | |
RUQXGVGYNKIGJD
|
7.8 | IC50 | 9 | — | |
XXTRJPVJIAZBBR
|
7.8 | IC50 | 2 | — | |
CCUMIOKJQCVBML
|
7.8 | IC50 | 2 | — | |
FBURYRMHEHTVED
|
7.8 | IC50 | 9 | — | |
JBWDTSLHUJHODF
|
7.8 | IC50 | 9 | — | |
OQSBQXVIMQMCES
|
7.8 | IC50 | 9 | — | |
UXUQVXDYXKMCGA
|
7.8 | Ki | 21 | — | |
VFLPOFHPMNYCOH
|
7.8 | IC50 | 7 | — | |
XNWKXXIGSPPPBH
|
7.8 | Ki | 31 | — | |
YGVLUDLFNRZMNT
|
7.8 | IC50 | 8 | — | |
YSBCFQVEEKUZSU
|
7.8 | IC50 | 7 | — | |
LQSUUCXGVOHOFM
|
7.8 | IC50 | 2 | — | |
NOAYWSNRHLCNJQ
|
7.8 | IC50 | 2 | — | |
PPALZSWDMRGSQV
|
7.8 | IC50 | 5 | — | |
JBWDTSLHUJHODF
|
7.8 | IC50 | 8 | — | |
OEVQTWCGWDOIFZ
|
7.8 | IC50 | 7 | — | |
OSWHZHVVVZAPRN
|
7.8 | IC50 | 6 | — | |
RLTCEYSNDOXWKS
|
7.8 | IC50 | 7 | — | |
SJWUVVGOTOMGOH
|
7.8 | IC50 | 10 | — | |
ITOTZLBIDAOTGK
|
7.8 | IC50 | 4 | — | |
SJYQOVMGZOATNK
|
7.8 | IC50 | 9 | — | |
ARYGGCNDASPYNG
|
7.7 | IC50 | 3 | — | |
ITOTZLBIDAOTGK
|
7.7 | IC50 | 4 | — | |
MOYYMSNZEWQWQJ
|
7.7 | IC50 | 3 | — | |
NFPDLDFOSLPKHQ
|
7.7 | IC50 | 2 | — | |
PINHQPCEXCQCGH
|
7.7 | IC50 | 2 | — | |
WAJNOEPHTZIWTO
|
7.7 | IC50 | 6 | — | |
ZYVXTMKTGDARKR
|
7.7 | IC50 | 6 | — | |
BWNXEFDIXGZHPQ
|
7.7 | IC50 | 4 | — | |
DXVSNYWBRDTHFF
|
7.7 | IC50 | 9 | — | |
KRXQWLCJHMDEDM
|
7.7 | IC50 | 8 | — | |
VAXXXDBEUYQWBN
|
7.7 | IC50 | 2 | — | |
CFBADDSSFSYJPF
|
7.7 | Ki | 23 | — | |
CLEGDJQQHUTCOW
|
7.7 | Ki | 43 | — | |
DKXHSOUZPMHNIZ
|
7.7 | Ki | 51 | Yes | |
DQPYZHUAILXFJI
|
7.7 | Ki | 27 | — | |
DYSRECIVMDGUQU
|
7.7 | Ki | 29 | — | |
GDYZFFBMSBDTAA
|
7.7 | Ki | 60 | — |