Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ORBNLRQBHQLUIW
|
8.0 | IC50 | 2 | — | |
OVVHFDIQCYTOAS
|
8.0 | IC50 | 9 | — | |
RFBPWKMQWSIPEO
|
8.0 | Ki | 28 | — | |
SLKCVFPEQGHNSI
|
8.0 | Ki | 29 | — | |
WCGVAQKYQAEAIH
|
8.0 | IC50 | 2 | — | |
XJJYJNMNYDNXNO
|
8.0 | Ki | 23 | — | |
YJKPCYDSZXIODK
|
8.0 | IC50 | 8 | — | |
YNGHSMIWDSRNCH
|
8.0 | IC50 | 2 | — | |
ZKLJKKASNXVQBZ
|
8.0 | Ki | 27 | — | |
ZYTFPHRVOZXPGZ
|
8.0 | Ki | 30 | — | |
HJEKFRDOAYXXRU
|
8.0 | IC50 | 8 | — | |
JQVRJDHSZIESJC
|
8.0 | IC50 | 2 | — | |
FOIOWDZKEWEOQP
|
8.0 | IC50 | 2 | — | |
GHQYHWMWJLSKRP
|
8.0 | IC50 | 9 | — | |
GUXARCGBVPDGMI
|
8.0 | IC50 | 3 | — | |
HQAFQRVIFUNAKT
|
8.0 | IC50 | 3 | — | |
IJFKKIMDRSZOOW
|
8.0 | IC50 | 8 | — | |
JXQZHHAAJMQJKU
|
8.0 | IC50 | 9 | — | |
UEFCSGDOOJJXTN
|
8.0 | IC50 | 46 | — | |
UZKITQOBTXEXSY
|
8.0 | IC50 | 2 | — | |
JNTIINGGIOJIMW
|
7.9 | IC50 | 4 | — | |
FUSZCAJFRIHBLV
|
7.9 | IC50 | 4 | — | |
AKNIGLLNHUTMPO
|
7.9 | IC50 | 9 | — | |
BGVLELSCIHASRV
|
7.9 | IC50 | 12 | — | |
BQALMWBXRVWKAM
|
7.9 | IC50 | 2 | — | |
GBNWWXHUOVAUHT
|
7.9 | IC50 | 4 | Yes | |
KUFCYNGJQRKYSQ
|
7.9 | IC50 | 2 | — | |
MXEZQEFCKXVMFN
|
7.9 | IC50 | 5 | — | |
QTRZNDLLYHSJSH
|
7.9 | IC50 | 9 | — | |
SDAAXACYZBWYTQ
|
7.9 | IC50 | 2 | — | |
SJWUVVGOTOMGOH
|
7.9 | IC50 | 9 | — | |
WREJZZXSNOJGIW
|
7.9 | IC50 | 8 | — | |
YHZQZEGQCKWCLP
|
7.9 | IC50 | 9 | — | |
LCHCSKHPVCDXAU
|
7.9 | Ki | 30 | — | |
LSLPDHNUWRDOGC
|
7.9 | Ki | 25 | — | |
XZONYYFHQICDAM
|
7.9 | Ki | 19 | — | |
AOGIFFVMTGMFBP
|
7.9 | IC50 | 8 | — | |
CIJWGWNHXQYIJC
|
7.9 | IC50 | 5 | — | |
CZWJLLBPWLUINU
|
7.9 | IC50 | 10 | — | |
DNJISDHVBHLOGY
|
7.9 | IC50 | 2 | — | |
JBWDTSLHUJHODF
|
7.9 | IC50 | 9 | — | |
RAQBQAXSLHDSKW
|
7.9 | IC50 | 8 | — | |
RLTCEYSNDOXWKS
|
7.9 | IC50 | 9 | — | |
VRGNMDTYOWQXQC
|
7.9 | IC50 | 8 | — | |
VRGNMDTYOWQXQC
|
7.9 | IC50 | 5 | — | |
KJCRALOGJOLXCU
|
7.9 | IC50 | 3 | — | |
WYEVMOFRKALLJA
|
7.9 | IC50 | 4 | — | |
PMDAVRLCSZSLRH
|
7.9 | IC50 | 13 | — | |
UBGUCDLLEIGHHP
|
7.9 | IC50 | 6 | — | |
ZLFXEVGPZWFVCB
|
7.9 | IC50 | 2 | — |