Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KIMRTWGQATWAQF
|
8.2 | IC50 | 2 | — | |
NMUDZNRXZXDYEQ
|
8.2 | IC50 | 9 | — | |
OGPJOAYIAOEJAM
|
8.2 | IC50 | 8 | — | |
OYDWEMSWMQKSLK
|
8.2 | IC50 | 8 | — | |
QCJWUXFCDRVWGH
|
8.2 | IC50 | 2 | — | |
SDRAETFVRBBLOB
|
8.2 | IC50 | 5 | — | |
UZIATSFXNVOVFE
|
8.2 | IC50 | 2 | — | |
FLEAYYMORDPWAJ
|
8.2 | Ki | 90 | — | |
KHGPYYFCIAISBU
|
8.2 | Ki | 31 | — | |
NGDNKYRUKIPCLK
|
8.2 | Ki | 12 | — | |
QTHCAAFKVUWAFI
|
8.2 | IC50 | 23 | — | |
UDFDIIVNIYWXDM
|
8.2 | Ki | 74 | — | |
XXSPHNFKLDJDAK
|
8.2 | Ki | 26 | — | |
CGECJCJUHCZZGO
|
8.2 | IC50 | 9 | — | |
PVFNDFZQGWYILU
|
8.2 | IC50 | 3 | — | |
MUOKSQABCJCOPU
|
8.2 | IC50 | 36 | — | |
CGRDYMCBGXJNLR
|
8.2 | IC50 | 9 | — | |
DCHAEDURAZJASA
|
8.2 | IC50 | 9 | — | |
NSDQDNNJFIKBKR
|
8.2 | IC50 | 6 | — | |
SLKHMZQUNIHINK
|
8.2 | IC50 | 10 | — | |
UMWJBFSPIYCGRG
|
8.2 | IC50 | 7 | — | |
BWRQNVDGLTUELI
|
8.1 | IC50 | 5 | — | |
ZDINVWCJHPMIKS
|
8.1 | IC50 | 2 | — | |
GCYXEGSPUDSZJY
|
8.1 | Ki | 82 | — | |
GHMRUNOHAHJNNA
|
8.1 | Ki | 29 | — | |
GHNZOLKSIZOQCZ
|
8.1 | IC50 | 2 | — | |
GRHRWVRWLAIBGN
|
8.1 | IC50 | 5 | — | |
IOUKAQLHORTKRT
|
8.1 | IC50 | 3 | — | |
JAJFJEDUYYFVEE
|
8.1 | IC50 | 2 | — | |
KAKGFGCTONHQJW
|
8.1 | Ki | 25 | — | |
MGEGGAFJSKMJJD
|
8.1 | IC50 | 5 | — | |
PVMYRLVGSWLCSL
|
8.1 | IC50 | 2 | — | |
UIVOWAUHPLCYNK
|
8.1 | IC50 | 2 | — | |
XPHWIERLJBFPFV
|
8.1 | Ki | 69 | — | |
LQLBWZJHRARWDB
|
8.1 | IC50 | 6 | — | |
HKCITBQBYLZFBK
|
8.1 | IC50 | 3 | — | |
JMENQRYRZLNDDO
|
8.1 | IC50 | 2 | — | |
ANKYADWZYKSCAJ
|
8.1 | IC50 | 7 | — | |
HAPIHWIYVZOFQR
|
8.1 | IC50 | 4 | — | |
SDSQMAISOKRJPN
|
8.1 | IC50 | 2 | — | |
UTGHIUITNUXCRZ
|
8.1 | IC50 | 2 | — | |
UTGHIUITNUXCRZ
|
8.1 | IC50 | 2 | — | |
YAXGFAAKCUOWNM
|
8.1 | IC50 | 9 | — | |
CLIWAKTWXZNUAC
|
8.0 | IC50 | 2 | — | |
PEXTWZUAIQCVBB
|
8.0 | IC50 | 3 | — | |
PUGXENIKUPHCAF
|
8.0 | IC50 | 3 | — | |
AAYFHKFUAWLHMY
|
8.0 | IC50 | 5 | — | |
ANBPRTXIECGGEM
|
8.0 | IC50 | 2 | — | |
CEFPPDKMUCDGCU
|
8.0 | IC50 | 3 | — | |
KHQYSWUSDRSLMP
|
8.0 | IC50 | 2 | — |