Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RDWOWHGVIKYPLI
|
8.6 | IC50 | 2 | — | |
DXVSNYWBRDTHFF
|
8.5 | IC50 | 10 | — | |
FIVWKNZKXNNFCW
|
8.5 | IC50 | 9 | — | |
NBTJWRPKGNQBJS
|
8.5 | IC50 | 8 | — | |
USYASDQVUTWEQM
|
8.5 | IC50 | 9 | — | |
WHPORTUXBLFUPA
|
8.5 | IC50 | 8 | — | |
WHPORTUXBLFUPA
|
8.5 | IC50 | 9 | — | |
YSODDCRKIDDXKM
|
8.5 | IC50 | 9 | — | |
YVQOYBIBWBAHKH
|
8.5 | IC50 | 12 | — | |
ADMFLILDQJSEIK
|
8.5 | Ki | 72 | — | |
BGYVWFZMYBWCNY
|
8.5 | Ki | 30 | — | |
LHQWPYOYDRVMFI
|
8.5 | Ki | 21 | — | |
LYADGAGFYYXXIO
|
8.5 | IC50 | 82 | — | |
YSBCFQVEEKUZSU
|
8.5 | IC50 | 9 | — | |
ZBELDPMWYXDLNY
|
8.4 | IC50 | 4 | — | |
ZGFYGZLBXCHRCV
|
8.4 | IC50 | 2 | — | |
FIVWKNZKXNNFCW
|
8.4 | IC50 | 8 | — | |
GWJHMRBQEUHFOC
|
8.4 | Ki | 42 | — | |
IVSYLIPATGYBCZ
|
8.4 | IC50 | 7 | — | |
ORUUEFDGYYTXAF
|
8.4 | Ki | 26 | — | |
OWFLADWRSCINST
|
8.4 | Ki | 30 | — | |
ROPFCXUWNMYMSW
|
8.4 | IC50 | 10 | — | |
UDGAFXWTODQSMC
|
8.4 | IC50 | 2 | — | |
XFWUTMHVDGPWLH
|
8.4 | Ki | 75 | — | |
YORVMWUGDVGXOQ
|
8.4 | IC50 | 8 | — | |
LTQMADLYBJVCSN
|
8.3 | IC50 | 2 | — | |
UZIATSFXNVOVFE
|
8.3 | IC50 | 9 | — | |
PTTXGLLPYLIZCU
|
8.3 | IC50 | 2 | — | |
QHTJZFWEQYRYQE
|
8.3 | IC50 | 9 | — | |
VCCCOYOXNKTQFO
|
8.3 | IC50 | 9 | — | |
HFJRGZBUEXFBMO
|
8.3 | IC50 | 2 | — | |
BBCSUMURJUYILA
|
8.3 | IC50 | 9 | — | |
BNPUEXLGIHXXJP
|
8.3 | IC50 | 2 | — | |
BULHRWBHKAVJMT
|
8.3 | IC50 | 8 | — | |
CWRTWFWDDAJOMG
|
8.3 | IC50 | 4 | Yes | |
DCJOTKUJWJFCSP
|
8.3 | IC50 | 9 | — | |
HKSZLNNOFSGOKW
|
8.3 | IC50 | 408 | — | |
MRWURALZVKJHPD
|
8.3 | IC50 | 2 | — | |
PBVAHEBIEXXNNA
|
8.3 | IC50 | 4 | — | |
PNKALLUVKOKYHZ
|
8.3 | Ki | 32 | — | |
SJWUVVGOTOMGOH
|
8.3 | IC50 | 12 | — | |
SKKBUBMBPCJYKW
|
8.3 | IC50 | 9 | — | |
SMRWVXLSRJWVBF
|
8.3 | Ki | 25 | — | |
UGYUFJPHSWYELP
|
8.3 | IC50 | 8 | — | |
URNZTLZSAVLTIZ
|
8.3 | Ki | 26 | — | |
QTRQYFCAAHDIDR
|
8.3 | IC50 | 2 | — | |
KYOPCGIPHGGWMV
|
8.3 | IC50 | 7 | — | |
LUKGZXVCOQQBHB
|
8.2 | IC50 | 2 | — | |
XQMMPFLQOCIGRW
|
8.2 | IC50 | 2 | — | |
GEJSQZULGDKBQV
|
8.2 | IC50 | 8 | — |