Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NRZYTPAJGVTKIM
|
6.3 | Ki | 38 | — | |
OROAFGSTGRDOFR
|
6.3 | Ki | 6 | — | |
PQNWNVWJXPSZFR
|
6.3 | Ki | 21 | — | |
UPITUWGOTMBQLX
|
6.3 | Ki | 13 | — | |
USSKXRGFNVFHFF
|
6.3 | IC50 | 7 | — | |
WICLISNBDMGFST
|
6.3 | Ki | 10 | — | |
ZCAOFAAOUBUUBJ
|
6.3 | Ki | 9 | — | |
BOLOCLITWRGHFA
|
6.3 | IC50 | 6 | — | |
GVANUSPDJMCBIK
|
6.3 | IC50 | 6 | — | |
IXTKPNOXAVTBCW
|
6.3 | IC50 | 4 | — | |
MXIKVRCYCKFUND
|
6.3 | IC50 | 6 | — | |
RVSPPVBZRQFLQY
|
6.3 | IC50 | 6 | — | |
FTZBKRUJACNIDE
|
6.3 | IC50 | 2 | — | |
QQFFZFFKGFYNKB
|
6.3 | IC50 | 2 | — | |
XUAFNTGABGAVRC
|
6.3 | IC50 | 2 | — | |
LGQKIASGYQMERJ
|
6.3 | IC50 | 3 | — | |
BWUOLNXJAQPJKF
|
6.2 | IC50 | 7 | — | |
HWDFAHKJNADKKP
|
6.2 | IC50 | 5 | — | |
KIUXCHKRJQPHFK
|
6.2 | IC50 | 4 | — | |
SJXZXKOJVKYIJT
|
6.2 | IC50 | 2 | — | |
XEFWAPMPJNMNEJ
|
6.2 | IC50 | 2 | — | |
DUQMBHQZRWIXEM
|
6.2 | IC50 | 2 | — | |
FJICMLZOGOVQRG
|
6.2 | IC50 | 4 | — | |
KQGHLDMPONJRNE
|
6.2 | IC50 | 3 | — | |
XNYOTZHBHJIMBV
|
6.2 | IC50 | 2 | — | |
BIDTZRBRWDXWHU
|
6.2 | IC50 | 2 | — | |
QNMZWFNNJMGJPU
|
6.2 | IC50 | 2 | — | |
XNWRZAZVQKFHKW
|
6.2 | IC50 | 2 | — | |
GQBQUBULFDQKBM
|
6.2 | IC50 | 4 | — | |
PKEDBIGNILOTHW
|
6.2 | IC50 | 2 | — | |
TVUWQDLBEOZVOU
|
6.2 | IC50 | 41 | — | |
UZLHPXPKYRQXJV
|
6.2 | IC50 | 2 | — | |
VTDMTVMKVZXVSP
|
6.2 | IC50 | 4 | — | |
AMHZZMGEDQCWKL
|
6.2 | IC50 | 4 | — | |
KZHOWDULHMQJNY
|
6.2 | IC50 | 2 | — | |
AOFJRBMLTUGMMP
|
6.2 | Ki | 12 | — | |
CBTNARFZVOPLBO
|
6.2 | IC50 | 5 | — | |
CTXSEYUOXKGIMM
|
6.2 | IC50 | 3 | — | |
DWHOVKRIZFMOSJ
|
6.2 | Ki | 4 | — | |
GXFGHUNNGNQSMQ
|
6.2 | Ki | 19 | — | |
IMHKMKWSWHFKTM
|
6.2 | Ki | 13 | — | |
JHYHWHUTTXJICB
|
6.2 | Ki | 18 | — | |
JMIIFJIJWDCOEP
|
6.2 | Ki | 15 | — | |
JOCUCEXJBMSIMH
|
6.2 | IC50 | 2 | — | |
KJFGBDYZIORKKA
|
6.2 | IC50 | 2 | — | |
MASJMHFQMYAPJR
|
6.2 | Ki | 41 | — | |
MZIOLOXGGOLJMJ
|
6.2 | Ki | 12 | — | |
OEEGUWWPGAZRIJ
|
6.2 | Ki | 21 | — | |
QNLMLEYLZSGBHP
|
6.2 | Ki | 8 | — | |
RYSOFKOEVPNDDI
|
6.2 | Ki | 9 | — |