Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IHGUHCPMDSTTIW
|
6.5 | Ki | 5 | — | |
IKEGFWWGERPFMP
|
6.5 | IC50 | 2 | — | |
JGBCLJZMLUMHOO
|
6.5 | Ki | 6 | — | |
KPVCGFZWGAYXMV
|
6.5 | Ki | 7 | — | |
KYACBMRLQMEIAI
|
6.5 | Ki | 30 | — | |
LRINYHMQZRENCY
|
6.5 | Ki | 29 | — | |
NSDIHUXUFJHXRA
|
6.5 | Ki | 11 | — | |
OEKYVFZKBRIDJO
|
6.5 | Ki | 12 | — | |
OETCTXGISYWYMV
|
6.5 | Ki | 7 | — | |
QDITZBLZQQZVEE
|
6.5 | Kd | 19 | — | |
SODGZPDNROVASD
|
6.5 | Ki | 7 | — | |
VWACUNWBMWWMPJ
|
6.5 | Ki | 18 | — | |
XGMWRIIMIJPGBH
|
6.5 | Ki | 10 | — | |
XLFYOIVELARSKP
|
6.5 | Ki | 33 | — | |
YEPNVBNYCRGZRX
|
6.5 | Ki | 26 | — | |
YYPKOMNJRZRWIC
|
6.5 | Ki | 26 | — | |
KVIRZIGSUYNQLP
|
6.5 | IC50 | 2 | — | |
YEFYCSKFDBXSSK
|
6.5 | IC50 | 7 | — | |
FSBMCTDYWXIBLM
|
6.5 | IC50 | 22 | — | |
LFSFZGXABLTIEJ
|
6.5 | IC50 | 3 | — | |
YWOJRGRRNWQSOH
|
6.5 | IC50 | 2 | — | |
CQZSVQKINMHLBO
|
6.5 | IC50 | 4 | — | |
HHUOQHKKRABAQB
|
6.5 | IC50 | 5 | — | |
OUSFTKFNBAZUKL
|
6.5 | Kd | 58 | Yes | |
OWEQZGPRBRSUEF
|
6.5 | IC50 | 2 | — | |
QGGNWMQODZFHNG
|
6.5 | IC50 | 4 | — | |
UXIAMCZUNQBRTJ
|
6.5 | IC50 | 4 | — | |
BUDHBLBYISRDCR
|
6.5 | IC50 | 2 | — | |
HMMICWRUNSZYCJ
|
6.5 | IC50 | 3 | — | |
NLNMWQUTXDGLJU
|
6.5 | IC50 | 5 | — | |
BZUXWEBTNNKFBN
|
6.5 | IC50 | 3 | — | |
FLWYCOJREJRWLJ
|
6.5 | IC50 | 3 | — | |
MGAHZVJVMCCAOO
|
6.4 | IC50 | 2 | — | |
CRVHQVJVMWGKAV
|
6.4 | IC50 | 3 | — | |
LKROTCXRJRCMTD
|
6.4 | IC50 | 4 | — | |
PAHHKMMVQJCPJI
|
6.4 | IC50 | 8 | — | |
LZUVHLORMNUQJL
|
6.4 | IC50 | 3 | — | |
NAYXGFSGXGZZCZ
|
6.4 | IC50 | 3 | — | |
VNRLVGZOAVIXDU
|
6.4 | IC50 | 4 | — | |
BULHRWBHKAVJMT
|
6.4 | IC50 | 8 | — | |
NKRFEKCLNDSTNO
|
6.4 | IC50 | 2 | — | |
OITUSVUYZAXFTD
|
6.4 | IC50 | 5 | — | |
VBYRFFCBZNEHAL
|
6.4 | IC50 | 4 | — | |
AQDWLHMFJHACCX
|
6.4 | Ki | 8 | — | |
ASRWRMWLFZMROI
|
6.4 | IC50 | 6 | — | |
ASRWRMWLFZMROI
|
6.4 | IC50 | 6 | — | |
BOSSBLQXHFNQIF
|
6.4 | IC50 | 3 | — | |
BZFGDXJGWSIYQP
|
6.4 | Ki | 9 | — | |
CZIGMBNEFWBEMD
|
6.4 | Ki | 16 | — | |
DCTBPIBEQFLAOQ
|
6.4 | Ki | 13 | — |