Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OWRXHGAFWZFFCW
|
6.6 | Ki | 113 | — | |
RFVBRKXQYUDGIO
|
6.6 | Ki | 23 | — | |
RPGBQFNDFPEOON
|
6.6 | Ki | 22 | — | |
UQJQNZHGEVLHST
|
6.6 | Ki | 15 | — | |
VQPBIJGXSXEOCU
|
6.6 | Ki | 24 | — | |
WCAKSXQRFBVWDG
|
6.6 | Ki | 10 | — | |
WZISGNDZZPSYRP
|
6.6 | Ki | 20 | — | |
XCHWBXBDZRJVDP
|
6.6 | Ki | 51 | — | |
ZCBUQCWBWNUWSU
|
6.6 | Kd | 59 | — | |
IDUYBYPYFGSSPE
|
6.6 | IC50 | 2 | — | |
IRBWROIEALHOPH
|
6.6 | IC50 | 7 | — | |
MXRBAJVBWGVZJI
|
6.6 | IC50 | 4 | — | |
NRHKUKQUEJSGMG
|
6.6 | IC50 | 3 | — | |
CTNPALGJUAXMMC
|
6.6 | Kd | 151 | — | |
FYRYKOQBRXRWER
|
6.6 | IC50 | 2 | — | |
IEFFSHLHNYVSEF
|
6.6 | IC50 | 8 | — | |
MNTINTDTQABOKE
|
6.6 | IC50 | 4 | — | |
NHHQJBCNYHBUSI
|
6.6 | Kd | 220 | — | |
ZJVGZWWTWGRGFK
|
6.6 | IC50 | 4 | — | |
FRPGBGWSLAGPND
|
6.6 | IC50 | 7 | — | |
YRFAWSIUIFNVQA
|
6.6 | IC50 | 4 | — | |
ZPKXDHHDZZKMKI
|
6.6 | IC50 | 6 | — | |
HFEVNTGRPXCJIM
|
6.5 | IC50 | 6 | — | |
JFIBFRPEOMMHJL
|
6.5 | IC50 | 2 | — | |
JQSJAVBMIMDUFO
|
6.5 | IC50 | 4 | — | |
QZIYOWZOZNSBGJ
|
6.5 | IC50 | 3 | — | |
UBUJLBVNZCRWPX
|
6.5 | IC50 | 7 | — | |
ZPKXDHHDZZKMKI
|
6.5 | IC50 | 6 | — | |
JZRNXAPRPJTGOG
|
6.5 | Kd | 3 | — | |
LHDIGZOUPVIOQB
|
6.5 | IC50 | 2 | — | |
PCHKPVIQAHNQLW
|
6.5 | IC50 | 8 | — | |
CROVEFPUGGIVBG
|
6.5 | IC50 | 2 | — | |
FQFGDUPFMGYOMB
|
6.5 | IC50 | 6 | — | |
IEJOMJUTRBOWNE
|
6.5 | Kd | 5 | — | |
KKVKVCZEAYHBCN
|
6.5 | IC50 | 2 | — | |
OSGPGSKNNFIBDD
|
6.5 | IC50 | 2 | — | |
PMXCMJLOPOFPBT
|
6.5 | IC50 | 17 | Yes | |
QSWUXXLUPIYCHQ
|
6.5 | IC50 | 2 | — | |
QVIIMXQIBJRPFS
|
6.5 | IC50 | 3 | — | |
SBNNOXYSSSCMJX
|
6.5 | IC50 | 6 | — | |
UJVJXKMEZMFCNM
|
6.5 | IC50 | 6 | — | |
VFLDPWHFBUODDF
|
6.5 | IC50 | 25 | — | |
VUEJIYSQTDBJDH
|
6.5 | IC50 | 2 | — | |
ABMAOGVUUQCYHD
|
6.5 | IC50 | 2 | — | |
HMDPCTZKMDHQTP
|
6.5 | IC50 | 5 | — | |
MHURZKJMJCNXDR
|
6.5 | IC50 | 5 | — | |
AWJPVXSHMIELNJ
|
6.5 | Ki | 23 | — | |
AXIVWWPYPSYJLD
|
6.5 | Ki | 7 | Yes | |
CACMTVGXYAZZNY
|
6.5 | Ki | 11 | — | |
DZIPQNPWTUXXSJ
|
6.5 | Ki | 18 | — |