Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RWAVDFHFFDMSHX
|
6.7 | IC50 | 4 | — | |
UMULGPSQNQMYNC
|
6.7 | Ki | 6 | — | |
UPPGGRZNGRFDAU
|
6.7 | Ki | 21 | — | |
UXVJSLNUZNAQHS
|
6.7 | IC50 | 2 | — | |
UZUFLDRZLTUMAC
|
6.7 | IC50 | 3 | — | |
VUDAXHCEPITOSW
|
6.7 | Ki | 4 | — | |
WINHZLLDWRZWRT
|
6.7 | Kd | 201 | Yes | |
WZSVRUCBLPTNFX
|
6.7 | Ki | 4 | — | |
XBDWKVLCDCUNHH
|
6.7 | Ki | 18 | — | |
YEHCNYAQEBQCCS
|
6.7 | Ki | 74 | — | |
YUOWJICKAJQZLS
|
6.7 | Ki | 35 | — | |
ZLVOTRRGLSDLPF
|
6.7 | Ki | 36 | — | |
CKKUHARWBUXFAW
|
6.7 | IC50 | 5 | — | |
GPMRASYSIQENIJ
|
6.7 | IC50 | 3 | — | |
DDJAQBRJAZWAAX
|
6.7 | IC50 | 4 | — | |
MOPUAJCKFRRYRF
|
6.7 | IC50 | 2 | — | |
MQJVDVMWBFSFHI
|
6.7 | IC50 | 5 | — | |
NKDOPEFRNJXAOV
|
6.7 | IC50 | 6 | — | |
WUJUMXFZYYLJKH
|
6.7 | IC50 | 2 | — | |
HEAGNKNMQVIVMM
|
6.7 | IC50 | 8 | — | |
HFYNRAVQEUKOFF
|
6.7 | IC50 | 3 | — | |
JTYIDARLAQQHPP
|
6.7 | IC50 | 4 | — | |
TYVKILZNVZGMIM
|
6.7 | IC50 | 2 | — | |
WKDIVCXCWMVLPY
|
6.7 | IC50 | 2 | — | |
YVSLJAICTSVCDB
|
6.7 | IC50 | 6 | — | |
AMUFSGPBIFOSNV
|
6.7 | IC50 | 3 | — | |
KQZBWTMAFLOSPA
|
6.7 | IC50 | 8 | — | |
SLPJGDQJLTYWCI
|
6.7 | IC50 | 6 | — | |
URXJBXVGNBGIJA
|
6.7 | IC50 | 5 | — | |
TWKWEBMGDALHPN
|
6.7 | IC50 | 9 | — | |
ZHTZVZJNJGCSJO
|
6.6 | IC50 | 7 | — | |
AKTCVLPOZVXXJU
|
6.6 | IC50 | 4 | — | |
RWUAJNWQCLQAAA
|
6.6 | IC50 | 4 | — | |
AXTAPYRUEKNRBA
|
6.6 | Kd | 24 | — | |
CEWIXDGUKGVYDQ
|
6.6 | IC50 | 7 | — | |
DVZORWAPBGBTCT
|
6.6 | IC50 | 4 | — | |
GCSZJMUFYOAHFY
|
6.6 | IC50 | 8 | — | |
GIQDYWGEMOCDSN
|
6.6 | IC50 | 5 | — | |
NZMFVJNZGKELJC
|
6.6 | IC50 | 4 | — | |
RUQXGVGYNKIGJD
|
6.6 | IC50 | 4 | — | |
IJELDUSMVKXTCW
|
6.6 | IC50 | 2 | — | |
ATGVCJYHNOSZEV
|
6.6 | Ki | 23 | — | |
BBZSEXSOPOXLIQ
|
6.6 | Ki | 8 | — | |
FGLPGUCHBHILNS
|
6.6 | Ki | 10 | — | |
GWXPHWSUMLUDPO
|
6.6 | Ki | 11 | — | |
HEUSUIRCBWROMH
|
6.6 | Ki | 64 | — | |
JFKIXRTUZAZONT
|
6.6 | Ki | 6 | — | |
OBZHLULOFFWAJX
|
6.6 | Ki | 8 | — | |
OHLKBSAOSZPTFS
|
6.6 | Ki | 9 | Yes | |
OKBNCPDNYVDCTG
|
6.6 | IC50 | 5 | — |