Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WYVDFOFDVCFARJ
|
6.9 | IC50 | 6 | — | |
YDTHCIZMSQZYMR
|
6.9 | IC50 | 7 | — | |
AEYLJTAIDDIOBA
|
6.9 | Ki | 53 | — | |
BQYDGSNDLAZAEW
|
6.9 | Ki | 13 | — | |
BWKADHBOXYDZFU
|
6.9 | IC50 | 10 | — | |
CLRFYTGANQZOBS
|
6.9 | Ki | 41 | — | |
DPSFKKBIIZTWDA
|
6.9 | IC50 | 3 | — | |
FDBPGAHVEGEARY
|
6.9 | Ki | 19 | — | |
GKODJBVKKLQMEY
|
6.9 | Ki | 10 | — | |
KRIUNPBAQZGFQA
|
6.9 | Ki | 76 | — | |
KRPDWHZTPZNLAZ
|
6.9 | IC50 | 5 | — | |
LDYVHYUGOBDUMZ
|
6.9 | IC50 | 6 | — | |
MPXAWSABMVLIBU
|
6.9 | IC50 | 6 | — | |
OPOGDZANLATWGS
|
6.9 | Ki | 9 | — | |
PAIFYAZSILXLBO
|
6.9 | Ki | 26 | — | |
QVLJVHWQAKYGQI
|
6.9 | IC50 | 8 | — | |
SLHUAYAGWNBZQC
|
6.9 | IC50 | 2 | — | |
VSVKFEMFAYXZKR
|
6.9 | Ki | 14 | Yes | |
XYZNKCSDQRKAFR
|
6.9 | Ki | 53 | — | |
ZFOMCSNUEHMROO
|
6.9 | IC50 | 7 | — | |
HUFHINCQVVFZJG
|
6.9 | IC50 | 2 | — | |
LELRIWOVACJYND
|
6.9 | IC50 | 5 | — | |
MEKFXUFACKZUCV
|
6.9 | IC50 | 9 | — | |
MWQLICNQHCLBLQ
|
6.9 | IC50 | 3 | — | |
NGFGTMFVWSDFPS
|
6.9 | IC50 | 32 | — | |
JLUXIHDOQQZMIZ
|
6.9 | IC50 | 4 | — | |
AOLMNCAPVYTEHC
|
6.9 | IC50 | 6 | — | |
CBZLUUYEFNCOHU
|
6.9 | IC50 | 2 | — | |
NWQZSQAVEPZDBP
|
6.9 | IC50 | 5 | — | |
YORVMWUGDVGXOQ
|
6.9 | IC50 | 8 | — | |
BHKVSOQUPYXVRZ
|
6.9 | IC50 | 6 | — | |
HHSNDNONCUTNQR
|
6.9 | IC50 | 7 | — | |
NVTNPVQFMSQPJQ
|
6.9 | IC50 | 7 | — | |
NXSJMRCTGYTSTK
|
6.9 | Kd | 200 | — | |
HFZLFYUNSURMIG
|
6.8 | IC50 | 3 | — | |
MIEPXFZAJZPNFG
|
6.8 | IC50 | 5 | — | |
MIEPXFZAJZPNFG
|
6.8 | IC50 | 8 | — | |
XMGLDSGFTZRJFY
|
6.8 | IC50 | 2 | — | |
YPTMZNNBDPEMOK
|
6.8 | IC50 | 6 | — | |
QVYXLOYBJBMXNP
|
6.8 | IC50 | 7 | — | |
XQQYRDDJENLAME
|
6.8 | IC50 | 8 | — | |
AWPWSWALRFFFFR
|
6.8 | IC50 | 2 | — | |
LMXLOYKFDZEHCS
|
6.8 | IC50 | 7 | — | |
BFZIDBAEKWSVSX
|
6.8 | IC50 | 5 | — | |
GFSFWVNETAIFJQ
|
6.8 | IC50 | 2 | — | |
PWBGPHVFGDQYNG
|
6.8 | IC50 | 3 | — | |
QTRZNDLLYHSJSH
|
6.8 | IC50 | 7 | — | |
WQYUNADCLFWKGN
|
6.8 | IC50 | 5 | — | |
WWRVEMKSOIGGCS
|
6.8 | IC50 | 5 | — | |
AXRCEOKUDYDWLF
|
6.8 | Kd | 31 | — |