Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LYNBNVBMAGDJRW
|
7.0 | Ki | 81 | — | |
MVRRAWJPZXNFMK
|
7.0 | IC50 | 6 | — | |
OHPRWVPOPFGLJG
|
7.0 | Ki | 19 | — | |
PHWHNHYZZNJPLB
|
7.0 | Ki | 16 | — | |
QATMNAAQTUISJK
|
7.0 | Ki | 13 | — | |
QCSOSYLYYAHPPY
|
7.0 | Ki | 2 | — | |
SHHUBFYLSRKFFE
|
7.0 | IC50 | 2 | — | |
UTFXYGYVDDLJER
|
7.0 | Ki | 36 | — | |
VVEGARMQKNYDID
|
7.0 | Ki | 24 | — | |
VWVYILCFSYNJHF
|
7.0 | Ki | 49 | — | |
WNKQZLFWZLQFOH
|
7.0 | IC50 | 3 | — | |
XZWVOUQIYLZUCJ
|
7.0 | Ki | 23 | — | |
YMIJUBCSOKSFRU
|
7.0 | Ki | 87 | — | |
ZGZVRPRSFXRGCF
|
7.0 | Ki | 76 | — | |
OSVUGUHRKMMBSE
|
7.0 | Kd | 170 | — | |
YRSCDRTXWYUNBB
|
7.0 | IC50 | 4 | Yes | |
CWJLAVRXVFHDSJ
|
7.0 | IC50 | 13 | — | |
RFOWEVIHKPOKTL
|
7.0 | IC50 | 4 | — | |
VGWCJGBQHCMHNJ
|
7.0 | IC50 | 8 | — | |
CXOICQRVGSVVHC
|
7.0 | IC50 | 2 | — | |
MFLKPCAUPXBTPC
|
7.0 | IC50 | 6 | — | |
QCZUWXJFWWURGI
|
7.0 | IC50 | 2 | — | |
SBZWDKFEGYDKIU
|
7.0 | IC50 | 2 | — | |
YKFHBMIPXGSMRS
|
7.0 | IC50 | 7 | — | |
AINKQRBPBUTJRM
|
7.0 | IC50 | 5 | — | |
CVDZJUNTQGTGHF
|
7.0 | IC50 | 4 | — | |
FTGAOPZDJRWUTG
|
7.0 | IC50 | 6 | — | |
HFLXYSRIPKXGOQ
|
7.0 | IC50 | 4 | — | |
UGHABJRZQKZAHP
|
7.0 | IC50 | 6 | — | |
UGUVGLVHRPLWRS
|
7.0 | IC50 | 3 | — | |
UGUVGLVHRPLWRS
|
7.0 | IC50 | 3 | — | |
DPIAIAIQEINUNP
|
7.0 | IC50 | 4 | — | |
XTJRKTBELWGSDN
|
7.0 | IC50 | 6 | — | |
MEZZCEDCBNWCRR
|
6.9 | IC50 | 7 | — | |
MYHMILRQDXANLR
|
6.9 | IC50 | 2 | — | |
KSSZBACUSMREEJ
|
6.9 | Ki | 2 | — | |
CKEWXVJUPNKAPF
|
6.9 | IC50 | 3 | — | |
DYIOAOFYWZXKEX
|
6.9 | IC50 | 4 | — | |
DYIOAOFYWZXKEX
|
6.9 | IC50 | 4 | — | |
JDNVNTCGESXSFD
|
6.9 | IC50 | 4 | — | |
KCTCLVINURCCIL
|
6.9 | IC50 | 6 | — | |
LZRHAZRGHSSHLR
|
6.9 | IC50 | 7 | — | |
MCNDTHVVURYHKT
|
6.9 | IC50 | 8 | — | |
OVPNQJVDAFNBDN
|
6.9 | Kd | 44 | Yes | |
PRJNNPMIUGYOST
|
6.9 | IC50 | 14 | — | |
RVYFLJXKEYHVBR
|
6.9 | IC50 | 5 | — | |
SDZHQRUPXPKDOD
|
6.9 | Ki | 2 | — | |
SZOYOCHRMSEEMG
|
6.9 | IC50 | 7 | — | |
WYQPGNJIFZHADC
|
6.9 | IC50 | 2 | — | |
CYEDYOVSORTFAY
|
6.9 | IC50 | 2 | — |