Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BIIVYFLTOXDAOV
|
7.1 | Kd | 82 | Yes | |
VOMDKRFMVUYOOQ
|
7.1 | IC50 | 4 | — | |
WSUWIXYPBRLNOT
|
7.1 | IC50 | 4 | — | |
BUDGLAJKNWCXIM
|
7.1 | IC50 | 4 | — | |
DYABBQVRJKEHMB
|
7.1 | IC50 | 2 | — | |
GCZJQTRRJPRFIP
|
7.1 | Ki | 10 | — | |
HOBMVEVXDIOMDM
|
7.1 | Ki | 18 | — | |
IUEBPIPDFMCSTP
|
7.1 | Ki | 29 | — | |
OHARPIGKJAKOCM
|
7.1 | IC50 | 8 | — | |
VBNPWXWJZJNXEY
|
7.1 | Ki | 18 | Yes | |
VHKRTWNLRWRPSB
|
7.1 | IC50 | 2 | — | |
WKWGFJFNCXAUEX
|
7.1 | Ki | 14 | Yes | |
YGVKOSRPXIWQPQ
|
7.1 | IC50 | 4 | — | |
YWITWZUKNXWOSD
|
7.1 | Ki | 10 | — | |
CBTNARFZVOPLBO
|
7.1 | IC50 | 8 | — | |
CHQYAWLKOUOTQO
|
7.1 | IC50 | 5 | — | |
OHNZJKJYATYGCV
|
7.1 | IC50 | 5 | — | |
GMWUNXLQEKAPBL
|
7.1 | IC50 | 2 | — | |
IEAUISSAHDPODS
|
7.1 | IC50 | 2 | — | |
IFLBFWBMAWIBBZ
|
7.1 | IC50 | 7 | — | |
QJVXFDORJYYPAW
|
7.1 | IC50 | 4 | — | |
SKAFXNGFXPGQIG
|
7.1 | Ki | 3 | — | |
XVVPNHZWUXCHJE
|
7.1 | IC50 | 3 | — | |
XDVWHWQSQJFRPP
|
7.1 | IC50 | 4 | — | |
IIGCQCAUAFMZHK
|
7.0 | Ki | 2 | — | |
SATMZMMKDDTOSQ
|
7.0 | IC50 | 2 | — | |
XDJCLCLBSGGNKS
|
7.0 | IC50 | 21 | — | |
CIEDQRFRRJHOSA
|
7.0 | IC50 | 6 | — | |
GCUNCFYJKLSBKK
|
7.0 | IC50 | 5 | — | |
OQGLPYHETIJRBX
|
7.0 | IC50 | 3 | — | |
OQGLPYHETIJRBX
|
7.0 | IC50 | 3 | — | |
QKCAXXVNZDAJAD
|
7.0 | IC50 | 5 | — | |
RVNDFXJEYCICIV
|
7.0 | IC50 | 7 | — | |
BEFUFKXGAMLMTP
|
7.0 | IC50 | 2 | — | |
DGSCWEKDRWDCOB
|
7.0 | IC50 | 5 | — | |
QLSWEZZOYCDEGC
|
7.0 | IC50 | 5 | — | |
ZCCPLJOKGAACRT
|
7.0 | Kd | 599 | — | |
ZSKIOUIBTZSAOT
|
7.0 | Ki | 2 | — | |
DCJGWITYNVWXGI
|
7.0 | IC50 | 2 | — | |
LGCHSPYDLIKTIC
|
7.0 | IC50 | 6 | — | |
PBJIOVQCYBRCRK
|
7.0 | IC50 | 5 | — | |
SIVLENRHVVVPKJ
|
7.0 | IC50 | 2 | — | |
XXIXFZAUCITSCM
|
7.0 | IC50 | 7 | — | |
BGVLELSCIHASRV
|
7.0 | Kd | 11 | — | |
BMGQWWVMWDBQGC
|
7.0 | Kd | 147 | Yes | |
DBKQWGCVGCVPIP
|
7.0 | Ki | 21 | — | |
DJUSDFVEBBYFFL
|
7.0 | Ki | 27 | — | |
HZCOFZVJMJRKIB
|
7.0 | IC50 | 2 | — | |
IJNGXROUMFEKDB
|
7.0 | Ki | 39 | — | |
LRLDYTTWQIFWBD
|
7.0 | Ki | 25 | — |