Target Details
| UniProt AC | Q13627 |
|---|---|
| Gene Symbol | DYRK1A |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,051
- Clinical molecules 24
- Avg pChEMBL 7.16
Associated Diseases (1)
Active Molecules (1,051)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GQQAKEHCSMJAKS
|
10.1 | Kd | 2 | — | |
DKZYXHCYPUVGAF
|
9.9 | Kd | 112 | — | |
KQVNWJXQFRWTDU
|
9.8 | Kd | 2 | — | |
NBMVLIXNQOYMFB
|
9.7 | Kd | 2 | — | |
QSGKPYRFWJINEH
|
9.7 | IC50 | 12 | — | |
WGNHFGLWDANFBX
|
9.6 | IC50 | 4 | — | |
JWEJSOFKTOSBBW
|
9.5 | IC50 | 4 | — | |
JGPBLWPUPCMPDV
|
9.5 | IC50 | 2 | — | |
RYBNARZBIXTFJS
|
9.4 | IC50 | 9 | — | |
RYBNARZBIXTFJS
|
9.4 | IC50 | 9 | — | |
ZPXSIWLYMMFFCE
|
9.4 | IC50 | 2 | — | |
OYVBBBNYTNSCKF
|
9.4 | IC50 | 2 | — | |
NWMPVMMGSHXANZ
|
9.4 | Ki | 58 | — | |
SRKBDTMNOSQJFR
|
9.2 | Kd | 2 | — | |
MNVPCONHWCXDES
|
9.2 | IC50 | 9 | — | |
ZKGOFDAUIALGLZ
|
9.1 | IC50 | 2 | — | |
ACSYKUPGCXYRRO
|
9.1 | Ki | 26 | — | |
RKUKAACYUCUJEE
|
9.1 | Ki | 58 | — | |
VONVAHFLRYRXSJ
|
9.0 | IC50 | 2 | — | |
AVKKQBJQERVCTD
|
9.0 | IC50 | 2 | — | |
BDMXFIMYKGLQAL
|
9.0 | IC50 | 9 | — | |
BUDHVVXPBGMAPV
|
9.0 | IC50 | 11 | — | |
BWNQBFHVFFZHMR
|
9.0 | IC50 | 10 | — | |
JFDRONLMXPRQPP
|
9.0 | IC50 | 9 | — | |
KHVQTEBOVFILCQ
|
9.0 | IC50 | 10 | — | |
LPILBMJJRGTKOQ
|
9.0 | Ki | 27 | — | |
PZRAWCBVDRNTDQ
|
9.0 | IC50 | 2 | — | |
QMUKOEKTUBVPFU
|
9.0 | IC50 | 12 | — | |
QXFBTYPBHYOEMX
|
9.0 | IC50 | 9 | — | |
RFRICXRVXVFZMF
|
9.0 | IC50 | 2 | — | |
VCTLOEWZYIGVBO
|
9.0 | IC50 | 12 | — | |
ZQVADOVUSXDTNV
|
9.0 | IC50 | 2 | — | |
HEVBCYZPXGZFGS
|
9.0 | IC50 | 11 | — | |
BGXZIBSLBRKDTP
|
8.9 | IC50 | 2 | — | |
OTKQTETZDVGXBV
|
8.8 | IC50 | 4 | — | |
BIMZUQRAGIDOLB
|
8.7 | IC50 | 2 | — | |
GXCOUFPTCZUTEE
|
8.7 | IC50 | 10 | — | |
BQWWOBKMDWACGC
|
8.7 | IC50 | 8 | — | |
CGPYAXSYKQBYKJ
|
8.7 | IC50 | 12 | — | |
CIICGXXZCWRFQE
|
8.7 | IC50 | 7 | — | |
KBMQGIPVJGXLOU
|
8.7 | IC50 | 7 | — | |
SBYPANVVFZBWDF
|
8.7 | IC50 | 9 | — | |
XCTYEZWILVGTGO
|
8.7 | IC50 | 9 | — | |
YEZMGVBTPDYRPO
|
8.7 | IC50 | 8 | — | |
BPNUQXPIQBZCMR
|
8.7 | Kd | 83 | Yes | |
JCJWCXBSDFGDSJ
|
8.7 | IC50 | 3 | — | |
CHQYAWLKOUOTQO
|
8.6 | IC50 | 20 | — | |
BSFNGHCTZDCQBF
|
8.6 | Ki | 93 | — | |
HKSZLNNOFSGOKW
|
8.6 | Ki | 118 | — | |
ZGGIYFOLDBTZIL
|
8.6 | Ki | 27 | — |