Target Details
| UniProt AC | Q13564 |
|---|---|
| Gene Symbol | NAE1 |
| Protein Name | NEDD8-activating enzyme E1 regulatory subunit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00899 (ThiF) |
Summary
- Multi-target molecules 127
- Clinical molecules 0
- Avg pChEMBL 7.01
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LAKZPZSUPYNBBK
|
6.3 | IC50 | 2 | — | |
LIJMFHOBJCEVMH
|
6.3 | IC50 | 2 | — | |
MCALKOUCNUORLI
|
6.3 | IC50 | 2 | — | |
MCALKOUCNUORLI
|
6.3 | IC50 | 2 | — | |
NDZNDPNVCPKYMJ
|
6.3 | IC50 | 2 | — | |
NLVWAWPOFPZCID
|
6.3 | IC50 | 2 | — | |
NVXDKPJHNLIHRT
|
6.3 | IC50 | 2 | — | |
PJBZQZVGHJDHCR
|
6.3 | IC50 | 2 | — | |
RBCSYQUJHUQLOM
|
6.3 | IC50 | 2 | — | |
RRQYUWVZNNLXLZ
|
6.3 | IC50 | 2 | — | |
SDTGWJVQSONSRT
|
6.3 | IC50 | 2 | — | |
UKZBRTAEEJPBDC
|
6.3 | IC50 | 2 | — | |
WSVVYAYWXLZXJS
|
6.3 | IC50 | 2 | — | |
XBPNVNABOVYYAV
|
6.3 | IC50 | 2 | — | |
ZVNMCNUGHPOVTE
|
6.3 | IC50 | 2 | — | |
CQPQXYFINJGAOR
|
6.3 | IC50 | 4 | — | |
STRXGXNXKPBKCD
|
6.3 | IC50 | 4 | — | |
LXRZVMYMQHNYJB
|
6.3 | IC50 | 4 | — | |
SPAPFFDHWAASPX
|
6.2 | IC50 | 4 | — | |
XKTWBXUBNVQZSI
|
6.2 | IC50 | 4 | — | |
SPZOHGTXTGPSCS
|
6.2 | IC50 | 4 | — | |
SRGSXTJJXYVFHF
|
6.2 | IC50 | 4 | — | |
AGIKMOLYLSSZIM
|
6.1 | IC50 | 4 | — | |
KIDRXSDFGBELIZ
|
6.1 | IC50 | 4 | — | |
SCTCXMGITXVTFZ
|
6.1 | IC50 | 4 | — | |
DOWYIWAYBWYUNF
|
6.0 | IC50 | 4 | — | |
LXRZVMYMQHNYJB
|
6.0 | IC50 | 6 | — |