Target Details
| UniProt AC | Q13564 |
|---|---|
| Gene Symbol | NAE1 |
| Protein Name | NEDD8-activating enzyme E1 regulatory subunit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00899 (ThiF) |
Summary
- Multi-target molecules 127
- Clinical molecules 0
- Avg pChEMBL 7.01
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HZGGNVPPVXVPMC
|
10.7 | IC50 | 2 | — | |
ZXVZEGZAHMZFDI
|
9.7 | IC50 | 2 | — | |
FRCOPIZAOPFHPW
|
9.3 | IC50 | 3 | — | |
LXRMIEAQCVCXPB
|
9.2 | IC50 | 2 | — | |
OVTMDKYPGLBLQS
|
9.2 | IC50 | 4 | — | |
GEVVUAXCPLJANF
|
9.1 | IC50 | 4 | — | |
TZTRUHFXPVXWRD
|
9.0 | IC50 | 4 | — | |
KRHLXBNCCSIYQF
|
8.7 | IC50 | 2 | — | |
LBCALMGKWJHMBW
|
8.6 | IC50 | 2 | — | |
FNWJTKORFPPIAM
|
8.6 | IC50 | 2 | — | |
NNCHFJOACARWTJ
|
8.4 | IC50 | 2 | — | |
MPUQHZXIXSTTDU
|
8.4 | IC50 | 3 | — | |
RRKVZTSURRTYAS
|
8.4 | IC50 | 2 | — | |
FYCFHQRHVRHJML
|
8.3 | IC50 | 4 | — | |
LVTJAGGEPATBEL
|
8.2 | IC50 | 2 | — | |
RXSJIXNVHKQDSE
|
8.2 | IC50 | 2 | — | |
SWSOEEHHAJZBIR
|
8.2 | IC50 | 2 | — | |
AXIJUIHSMBCUGV
|
8.1 | IC50 | 4 | — | |
IATSQDNCRGSWGA
|
8.0 | IC50 | 2 | — | |
GSIDFCOQKJFHGK
|
8.0 | IC50 | 2 | — | |
HKSXLMUAZXOPJU
|
8.0 | IC50 | 2 | — | |
PGAMXUGSHMQFKD
|
8.0 | IC50 | 3 | — | |
RSAMFWNUOBWHFF
|
8.0 | IC50 | 4 | — | |
ZKRPPCXDNMNUFZ
|
7.9 | IC50 | 2 | — | |
OXOQCSFIVOZOEF
|
7.9 | IC50 | 2 | — | |
ICGVNCCUMBPAKP
|
7.8 | IC50 | 2 | — | |
YCGZEMSJVAIEDZ
|
7.8 | IC50 | 2 | — | |
HUSXUHAWHWEADE
|
7.7 | IC50 | 4 | — | |
LYVXDBIEQKGPTI
|
7.7 | IC50 | 2 | — | |
NLFWBXFVORQEPK
|
7.7 | IC50 | 2 | — | |
NSRYFRUKRQLHSU
|
7.7 | IC50 | 2 | — | |
UWTVTBUAJYQNJJ
|
7.7 | IC50 | 4 | — | |
NLYVIEPYNMFUDJ
|
7.6 | IC50 | 4 | — | |
IZPAOFVHNJWLSN
|
7.5 | IC50 | 2 | — | |
IZYVMHSGDZFGFW
|
7.5 | IC50 | 4 | — | |
MTKDHLHKUOHZHT
|
7.5 | IC50 | 4 | — | |
WMFPYJXJTLDGIG
|
7.5 | IC50 | 4 | — | |
ZPRXBLNQGBGAAZ
|
7.4 | IC50 | 2 | — | |
PKHLGIWBWMPLAR
|
7.2 | IC50 | 4 | — | |
RQYBHYVLXAGXKU
|
7.2 | IC50 | 4 | — | |
QYTQASAQCLQDAW
|
7.2 | IC50 | 2 | — | |
FRVKNLCUOXIYII
|
7.1 | IC50 | 2 | — | |
VARKRXJNUKYOEA
|
7.1 | IC50 | 2 | — | |
JUVWGUHJFQQESY
|
7.0 | IC50 | 4 | — | |
SADMDVJVSZEYAB
|
7.0 | IC50 | 2 | — | |
AGIKMOLYLSSZIM
|
7.0 | IC50 | 4 | — | |
SSWIRGSVVTWUMX
|
7.0 | IC50 | 4 | — | |
RFDHMTHFEKUKQV
|
7.0 | IC50 | 2 | — | |
ZCKFJAREHQZZOB
|
7.0 | IC50 | 4 | — | |
UBPMFDHRGACICG
|
6.9 | IC50 | 2 | — |